Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50016513
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595424BDBM50595424(CHEMBL5172865)
Affinity DataKi:  0.00398nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595404BDBM50595404(CHEMBL5184455)
Affinity DataKi:  0.0200nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595423BDBM50595423(CHEMBL5190387)
Affinity DataKi:  0.0251nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595426BDBM50595426(CHEMBL5193853)
Affinity DataKi:  0.0251nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595427BDBM50595427(CHEMBL5200887)
Affinity DataKi:  0.0251nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595403BDBM50595403(CHEMBL5208201)
Affinity DataKi:  0.0398nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595405BDBM50595405(CHEMBL5184598)
Affinity DataKi:  0.0501nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595425BDBM50595425(CHEMBL5208957)
Affinity DataKi:  0.0501nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595403BDBM50595403(CHEMBL5208201)
Affinity DataIC50: 0.0501nMAssay Description:Invivo agonist beta2 adrenoceptor activity in Dunkin-Hartley guinea pig trachea assessed as histamine induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595423BDBM50595423(CHEMBL5190387)
Affinity DataKi:  0.0631nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595424BDBM50595424(CHEMBL5172865)
Affinity DataKi:  0.0631nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595424BDBM50595424(CHEMBL5172865)
Affinity DataIC50: 0.0794nMAssay Description:Invivo agonist beta2 adrenoceptor activity in Dunkin-Hartley guinea pig trachea assessed as histamine induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595426BDBM50595426(CHEMBL5193853)
Affinity DataKi:  0.0794nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595404BDBM50595404(CHEMBL5184455)
Affinity DataIC50: 0.100nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595404BDBM50595404(CHEMBL5184455)
Affinity DataIC50: 0.100nMAssay Description:Invivo agonist beta2 adrenoceptor activity in Dunkin-Hartley guinea pig trachea assessed as histamine induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595426BDBM50595426(CHEMBL5193853)
Affinity DataIC50: 0.126nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50569301BDBM50569301(CHEMBL4854091)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595404BDBM50595404(CHEMBL5184455)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595425BDBM50595425(CHEMBL5208957)
Affinity DataKi:  0.158nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595423BDBM50595423(CHEMBL5190387)
Affinity DataIC50: 0.158nMAssay Description:Invivo agonist beta2 adrenoceptor activity in Dunkin-Hartley guinea pig trachea assessed as histamine induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595424BDBM50595424(CHEMBL5172865)
Affinity DataIC50: 0.200nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595403BDBM50595403(CHEMBL5208201)
Affinity DataIC50: 0.200nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595427BDBM50595427(CHEMBL5200887)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50569301BDBM50569301(CHEMBL4854091)
Affinity DataKi:  0.251nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595403BDBM50595403(CHEMBL5208201)
Affinity DataKi:  0.316nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595425BDBM50595425(CHEMBL5208957)
Affinity DataIC50: 0.398nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595426BDBM50595426(CHEMBL5193853)
Affinity DataIC50: 0.398nMAssay Description:Invivo agonist beta2 adrenoceptor activity in Dunkin-Hartley guinea pig trachea assessed as histamine induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595425BDBM50595425(CHEMBL5208957)
Affinity DataIC50: 0.398nMAssay Description:Invivo agonist beta2 adrenoceptor activity in Dunkin-Hartley guinea pig trachea assessed as histamine induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595423BDBM50595423(CHEMBL5190387)
Affinity DataIC50: 0.501nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595405BDBM50595405(CHEMBL5184598)
Affinity DataIC50: 0.501nMAssay Description:Invivo agonist beta2 adrenoceptor activity in Dunkin-Hartley guinea pig trachea assessed as histamine induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595405BDBM50595405(CHEMBL5184598)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595406BDBM50595406(CHEMBL5200448)
Affinity DataKi:  0.794nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595427BDBM50595427(CHEMBL5200887)
Affinity DataIC50: 0.794nMAssay Description:Invivo agonist beta2 adrenoceptor activity in Dunkin-Hartley guinea pig trachea assessed as histamine induced contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595422BDBM50595422(CHEMBL5177499)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595408BDBM50595408(CHEMBL5195203)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595427BDBM50595427(CHEMBL5200887)
Affinity DataIC50: 2nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595416BDBM50595416(CHEMBL5178217)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595418BDBM50595418(CHEMBL5179380)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595419BDBM50595419(CHEMBL5194569)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595414BDBM50595414(CHEMBL5187593)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595420BDBM50595420(CHEMBL5193776)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595415BDBM50595415(CHEMBL5202045)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor(Guinea pig)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595405BDBM50595405(CHEMBL5184598)
Affinity DataIC50: 7.90nMAssay Description:Invivo antagonist activity at muscarinic M3 receptor activity in Dunkin-Hartley guinea pig trachea assessed as inhibition of carbachol induced contra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595409BDBM50595409(CHEMBL5202567)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595410BDBM50595410(CHEMBL5202787)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595413BDBM50595413(CHEMBL5195224)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595412BDBM50595412(CHEMBL5181855)
Affinity DataKi:  7.90nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595417BDBM50595417(CHEMBL5207792)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595429BDBM50595429(CHEMBL5201712)
Affinity DataKi:  25nMAssay Description:Displacement of 125I-cyanopindolol from human beta2 adrenoceptor expressed in CHO-K1 cell membrane measured after 1 hr by Cheng-prusoff equation anal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Chiesi Farmaceutici

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595407BDBM50595407(CHEMBL5193865)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-methylscopolamine from human muscarinic M3 receptor expressed in CHO-K1 cell membrane measured after 2 hr by Cheng-prusoff equat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details Article
PubMed
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