Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50019931
TargetMu-type opioid receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50624754(CHEMBL5400535)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]-Diprenorphine from human MOR receptor expressed in CHO-K1 cells assessed as inhibition constant measured for 1 hr by liquid scin...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNociceptin receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-Nociceptin from human NOP receptor expressed in CHO-K1 cells assessed as inhibition constant measured for 1 hr by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50624754(CHEMBL5400535)
Affinity DataKi: >1nMAssay Description:Displacement of [3H]-Diprenorphine from human DOR receptor expressed in CHO-K1 cells assessed as inhibition constant measured for 1 hr by liquid scin...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetMu-type opioid receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50019056(2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]-Diprenorphine from human MOR receptor expressed in CHO-K1 cells assessed as inhibition constant measured for 1 hr by liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetNociceptin receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50624754(CHEMBL5400535)
Affinity DataKi:  650nMAssay Description:Displacement of [3H]-Nociceptin from human NOP receptor expressed in CHO-K1 cells assessed as inhibition constant measured for 1 hr by liquid scintil...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM21025([D-Ala2-D-Leu5]enkephalin | (D-Ala2,D-Leu5)-Enkeph...)
Affinity DataKi:  1.07E+4nMAssay Description:Displacement of [3H]-Diprenorphine from human DOR receptor expressed in CHO-K1 cells assessed as inhibition constant measured for 1 hr by liquid scin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed