Compile Data Set for Download or QSAR
Report error Found 85 Enz. Inhib. hit(s) with all data for entry = 50020121
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626394(CHEMBL5431833)
Affinity DataIC50: 240nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626394(CHEMBL5431833)
Affinity DataIC50: 300nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626391(CHEMBL5411975)
Affinity DataIC50: 510nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626399(CHEMBL5439894)
Affinity DataIC50: 620nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626391(CHEMBL5411975)
Affinity DataIC50: 640nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626390(CHEMBL5414143)
Affinity DataIC50: 660nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626400(CHEMBL5435025)
Affinity DataIC50: 720nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626393(CHEMBL5409544)
Affinity DataIC50: 770nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626392(CHEMBL5435639)
Affinity DataIC50: 780nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626393(CHEMBL5409544)
Affinity DataIC50: 780nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626396(CHEMBL5400204)
Affinity DataIC50: 800nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626400(CHEMBL5435025)
Affinity DataIC50: 800nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626396(CHEMBL5400204)
Affinity DataIC50: 830nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626399(CHEMBL5439894)
Affinity DataIC50: 900nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626390(CHEMBL5414143)
Affinity DataIC50: 900nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626392(CHEMBL5435639)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626397(CHEMBL5440797)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626389(CHEMBL5432311)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626397(CHEMBL5440797)
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626389(CHEMBL5432311)
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626395(CHEMBL5419237)
Affinity DataIC50: 1.42E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626398(CHEMBL5405537)
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626398(CHEMBL5405537)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626395(CHEMBL5419237)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626363(CHEMBL5424895)
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626388(CHEMBL5394840)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626388(CHEMBL5394840)
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626363(CHEMBL5424895)
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626377(CHEMBL5424207)
Affinity DataIC50: 2.23E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626385(CHEMBL5420313)
Affinity DataIC50: 2.47E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626373(CHEMBL5432760)
Affinity DataIC50: 2.86E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626385(CHEMBL5420313)
Affinity DataIC50: 2.86E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626387(CHEMBL5440150)
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626357(CHEMBL5437305)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626384(CHEMBL5403879)
Affinity DataIC50: 3.22E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626387(CHEMBL5440150)
Affinity DataIC50: 3.23E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626383(CHEMBL5415469)
Affinity DataIC50: 3.62E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626386(CHEMBL5396885)
Affinity DataIC50: 3.86E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626359(CHEMBL5435156)
Affinity DataIC50: 3.87E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626362(CHEMBL5401812)
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626356(CHEMBL5429382)
Affinity DataIC50: 4.22E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626360(CHEMBL5406544)
Affinity DataIC50: 4.27E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626368(CHEMBL5397570)
Affinity DataIC50: 4.38E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626374(CHEMBL5431086)
Affinity DataIC50: 4.45E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626368(CHEMBL5397570)
Affinity DataIC50: 4.45E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626386(CHEMBL5396885)
Affinity DataIC50: 4.47E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626357(CHEMBL5437305)
Affinity DataIC50: 4.47E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626365(CHEMBL5430358)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626380(CHEMBL5397432)
Affinity DataIC50: 5.11E+3nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) using SGRGK(Ac)GGK(Ac)GLGK(Ac) GGAK(Ac)RHRK-biotinylated peptide as substrate incubated for 60 mins by alpha ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50626358(CHEMBL5412097)
Affinity DataIC50: 5.13E+3nMAssay Description:Inhibition of N-terminal GST-tagged/C-terminal 6His-tagged BRD4 BD1 (47 to 170 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
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