Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50018045
TargetCyclin-dependent kinase 9(Human)
Tongji University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50140257(CHEMBL16171 | 5,7-Dihydroxy-8-methoxy-2-phenyl-chr...)
Affinity DataIC50: 190nMAssay Description:Inhibition of CDK9 (unknown origin) using [33-p]-ATP as substrate incubated for 40 mins by Western blot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetE3 ubiquitin-protein ligase RNF114(Human)
Tongji University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50607224(CHEMBL5218793)
Affinity DataIC50: 240nMAssay Description:Inhibition of RNF114 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Human)
Tongji University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50607226(CHEMBL5220731)
Affinity DataIC50: 250nMAssay Description:Inhibition of HMGCR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetCyclin-dependent kinase 9(Human)
Tongji University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50607227(CHEMBL4530229)
Affinity DataIC50: 523nMAssay Description:Inhibition of CDK9 (unknown origin) incubated for 1 hr by fluorescent polarisation based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
Target3-hydroxy-3-methylglutaryl-coenzyme A reductase(Human)
Tongji University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50607225(CHEMBL5218794)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of HMGCR (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed