Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50018778
Affinity DataEC50: 3.30E+4nMAssay Description:Inhibition of human PGAM1 in human MDA-MB-231 cells assessed as decrease in PGAM1 activity incubated for 2 hrs by UV/Vis spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKd: 7.20E+3nMAssay Description:Binding affinity to PGAM1 (unknown origin) assessed as dissociation constant by fluorescence-based assayMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 105nMAssay Description:Inhibition of recombinant PGAM1 (unknown origin) assessed as decrease in absorbance in presence of LDH, pyruvate kinase M2 and NADH by spectroscopic ...More data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant PGAM1 (unknown origin) assessed as decrease in absorbance in presence of LDH, pyruvate kinase M2 and NADH by spectroscopic ...More data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Inhibition of His-tagged recombinant PGAM1 (unknown origin) assessed as reduction in ATP production in presence of pyruvate kinase M1 and ATP by Kina...More data for this Ligand-Target Pair
Affinity DataIC50: 770nMAssay Description:Inhibition of recombinant PGAM1 (unknown origin) assessed as decrease in absorbance in presence of LDH, pyruvate kinase M2 and NADH by spectroscopic ...More data for this Ligand-Target Pair
Affinity DataIC50: 850nMAssay Description:Allosteric inhibition of PGAM1 (unknown origin) assessed as decrease in absorbance in presence of LDH, pyruvate kinase M2 and NADH by spectroscopic a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of His-tagged recombinant PGAM1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in absorbance from oxidation of N...More data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of His-tagged recombinant PGAM1 (unknown origin) expressed in Escherichia coli BL21 assessed as decrease in absorbance from oxidation of N...More data for this Ligand-Target Pair
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of recombinant PGAM1 (unknown origin) assessed as decrease in absorbance in presence of LDH, pyruvate kinase M2 and NADH by spectroscopic ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of His6-tagged human PGAM1 expressed in Escherichia coli BL21(DE3)pLysS cells assessed as decrease in autofluorescence from oxidation of N...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of His6-tagged human PGAM1 expressed in Escherichia coli BL21(DE3)pLysS cells assessed as decrease in autofluorescence from oxidation of N...More data for this Ligand-Target Pair
