Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50020736
TargetFibroblast growth factor receptor 1(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 2579BDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 34nMAssay Description:Inhibition of FGFR-1 (unknown origin) incubated for 60 mins in presence of ATP by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5446BDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 37nMAssay Description:Inhibition of recombinant EGFR (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 16673BDBM16673(BAY439006 | CHEMBL1336 | BAY 43-9006 | 4-[4-({[4-c...)
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633199BDBM50633199(CHEMBL5398753)
Affinity DataIC50: 66nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetFibroblast growth factor receptor 1(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633199BDBM50633199(CHEMBL5398753)
Affinity DataIC50: 82nMAssay Description:Inhibition of FGFR-1 (unknown origin) incubated for 60 mins in presence of ATP by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50595124BDBM50595124(VANDETANIB | CHEBI:49960 | Vandetanib | GNF-PF-218...)
Affinity DataIC50: 94nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633199BDBM50633199(CHEMBL5398753)
Affinity DataIC50: 98nMAssay Description:Inhibition of recombinant EGFR (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633204BDBM50633204(CHEMBL5395205)
Affinity DataIC50: 108nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633202BDBM50633202(CHEMBL5404512)
Affinity DataIC50: 146nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633200BDBM50633200(CHEMBL5415189)
Affinity DataIC50: 242nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633203BDBM50633203(CHEMBL5402749)
Affinity DataIC50: 438nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633205BDBM50633205(CHEMBL5396585)
Affinity DataIC50: 455nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
National Center for Radiation Research and Technology (NCRRT)

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50633201BDBM50633201(CHEMBL5399404)
Affinity DataIC50: 536nMAssay Description:Inhibition of recombinant VEGFR2 (unknown origin) by kinase glo detection reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed