Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50015867
TargetCannabinoid receptor 2(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50590160(CHEMBL5172277)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of accumulation of forskolin-stimulated cAMP level incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50006250(CHEMBL3139186)
Affinity DataEC50:  49nMAssay Description:Agonist activity at human CB2 receptor expressed in PathHunter CHO-K1 CNR2 beta-arrestin cells assessed as beta-arrestin recruitment incubated for 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  58nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of accumulation of forskolin-stimulated cAMP level incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50006250(CHEMBL3139186)
Affinity DataEC50:  69nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of accumulation of forskolin-stimulated cAMP level incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50590159(CHEMBL5208097)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as inhibition of accumulation of forskolin-stimulated cAMP level incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataEC50:  164nMAssay Description:Agonist activity at human CB2 receptor expressed in PathHunter CHO-K1 CNR2 beta-arrestin cells assessed as beta-arrestin recruitment incubated for 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50590160(CHEMBL5172277)
Affinity DataEC50:  167nMAssay Description:Agonist activity at human CB2 receptor expressed in PathHunter CHO-K1 CNR2 beta-arrestin cells assessed as beta-arrestin recruitment incubated for 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Arrival Discovery

Curated by ChEMBL
LigandPNGBDBM50590159(CHEMBL5208097)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human CB2 receptor expressed in PathHunter CHO-K1 CNR2 beta-arrestin cells assessed as beta-arrestin recruitment incubated for 3 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed