Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50019160
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349534(CHEMBL5419465)
Affinity DataIC50: 0.230nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349535(CHEMBL5399511)
Affinity DataIC50: 0.290nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349533(CHEMBL5422048)
Affinity DataIC50: 0.380nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349536(CHEMBL5425432)
Affinity DataIC50: 0.910nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349537(CHEMBL5434099)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475762(CHEMBL5407216)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50475761(CHEMBL5414818)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50420241(CHEMBL5416221)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349537(CHEMBL5434099)
Affinity DataEC50:  5nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349527(CHEMBL5417798)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349537(CHEMBL5434099)
Affinity DataIC50: 6.10nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349531(CHEMBL5403188)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349530(CHEMBL5427454)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349532(CHEMBL5397546)
Affinity DataIC50: 16nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349528(CHEMBL5397310)
Affinity DataIC50: 16nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349529(CHEMBL5405297)
Affinity DataIC50: 27nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349526(CHEMBL5414505)
Affinity DataIC50: 84nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349524(CHEMBL5400561)
Affinity DataIC50: 167nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349525(CHEMBL5422617)
Affinity DataIC50: 474nMAssay Description:Inhibition of Escherichia coli FabH expressed in Escherichia coli DH10B cells assessed as incorporation of 3H signal in the product after 25 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
LigandPNGBDBM50349533(CHEMBL5422048)
Affinity DataIC50: 1.80E+3nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
LigandPNGBDBM50349534(CHEMBL5419465)
Affinity DataIC50: 6.10E+3nMAssay Description:Compound was tested for Adrenergic activity against Alpha-2 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
LigandPNGBDBM50349535(CHEMBL5399511)
Affinity DataIC50: 1.30E+4nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-1 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
LigandPNGBDBM50475762(CHEMBL5407216)
Affinity DataIC50: 2.40E+4nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
LigandPNGBDBM50349530(CHEMBL5427454)
Affinity DataIC50: 2.40E+4nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-1 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
LigandPNGBDBM50349537(CHEMBL5434099)
Affinity DataIC50: 2.90E+4nMAssay Description:Compound was evaluated for Adrenergic activity in Alpha-2 adrenergic receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetMonocarboxylate transporter 1(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50349537(CHEMBL5434099)
Affinity DataIC50: 3.00E+4nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-1 adrenergic receptor from rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
LigandPNGBDBM50420241(CHEMBL5416221)
Affinity DataIC50: 3.30E+4nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
LigandPNGBDBM50475761(CHEMBL5414818)
Affinity DataIC50: 3.30E+4nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
LigandPNGBDBM50349536(CHEMBL5425432)
Affinity DataIC50: 3.30E+4nMAssay Description:Compound was evaluated for Adrenergic activity against Alpha-2 adrenergic receptor in human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed