Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50019972
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625234(CHEMBL5415225)
Affinity DataIC50: 7nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625219(CHEMBL5396169)
Affinity DataIC50: 17nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625220(CHEMBL5416007)
Affinity DataIC50: 17nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625218(CHEMBL5396294)
Affinity DataIC50: 19nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625235(CHEMBL5439210)
Affinity DataIC50: 19nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625232(CHEMBL5399021)
Affinity DataIC50: 24nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625217(CHEMBL5419657)
Affinity DataIC50: 24nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625237(CHEMBL5415283)
Affinity DataIC50: 25nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625216(CHEMBL5416991)
Affinity DataIC50: 27nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625233(CHEMBL5433686)
Affinity DataIC50: 32nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625211(CHEMBL5428990)
Affinity DataIC50: 34nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625230(CHEMBL5396133)
Affinity DataIC50: 36nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625210(CHEMBL5394045)
Affinity DataIC50: 36nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM109086(US8604016, 670 | US9938267, Cmpd ID 670 | US107935...)
Affinity DataIC50: 52nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625231(CHEMBL5399039)
Affinity DataIC50: 68nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625205(CHEMBL5428837)
Affinity DataIC50: 79nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625204(CHEMBL5429833)
Affinity DataIC50: 87nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625203(CHEMBL5412557)
Affinity DataIC50: 110nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625215(CHEMBL5423461)
Affinity DataIC50: 130nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625206(CHEMBL5411562)
Affinity DataIC50: 140nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625229(CHEMBL5414772)
Affinity DataIC50: 160nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625212(CHEMBL5417938)
Affinity DataIC50: 170nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625213(CHEMBL5437177)
Affinity DataIC50: 190nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625214(CHEMBL5436876)
Affinity DataIC50: 220nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625208(CHEMBL5411575)
Affinity DataIC50: 240nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625201(CHEMBL5411945)
Affinity DataIC50: 280nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625224(CHEMBL5415915)
Affinity DataIC50: 290nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625223(CHEMBL5409568)
Affinity DataIC50: 390nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625225(CHEMBL5422173)
Affinity DataIC50: 520nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625202(CHEMBL5396896)
Affinity DataIC50: 530nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625222(CHEMBL5427008)
Affinity DataIC50: 580nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625221(CHEMBL5405118)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625207(CHEMBL5397662)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625209(CHEMBL5411598)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625228(CHEMBL5393992)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625236(CHEMBL5430383)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625226(CHEMBL5411235)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetGlutaminase kidney isoform, mitochondrial(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625227(CHEMBL5432785)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of GLS1 (unknown origin) preincubated for 10 mins followed by glutamine addition measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed