Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 50018611
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50064751(CHEMBL3403780)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
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TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554975(CHEMBL4595209)
Affinity DataKi:  224nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50065915(CHEMBL3401461)
Affinity DataKi:  277nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50610306(CHEMBL5285428)
Affinity DataKi:  487nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50064645(CHEMBL3403768)
Affinity DataKi:  612nMAssay Description:Displacement of [3H]RTI-33 from GPR88 (unknown origin) by competition binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM50554975(CHEMBL4595209)
Affinity DataKd:  41nMAssay Description:Binding affinity to GPR88 in mouse striatal membrane by filtration methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50064751(CHEMBL3403780)
Affinity DataEC50:  304nMAssay Description:Agonist activity at GPR88 (unknown origin) transfected in HEK293 cells assessed as cAMP level by GloSensor cAMP assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50610306(CHEMBL5285428)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at GPR88 (unknown origin) transfected in HEK293 cells assessed as cAMP level by GloSensor cAMP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50065915(CHEMBL3401461)
Affinity DataEC50:  74nMAssay Description:Agonist activity at GPR88 (unknown origin) transfected in HEK293 cells assessed as cAMP level by GloSensor cAMP assayMore data for this Ligand-Target Pair
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554975(CHEMBL4595209)
Affinity DataEC50:  45nMAssay Description:Agonist activity at GPR88 (unknown origin) transfected in HEK293 cells assessed as cAMP level by GloSensor cAMP assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50554975(CHEMBL4595209)
Affinity DataKd:  85nMAssay Description:Binding affinity to PPLS-HA tagged human GPR88 expressed in CHO cell membrane by filtration methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProbable G-protein coupled receptor 88(Homo sapiens (Human))TBA
LigandPNGBDBM50064645(CHEMBL3403768)
Affinity DataEC50:  195nMAssay Description:Agonist activity at GPR88 (unknown origin) transfected in HEK293 cells assessed as cAMP level by GloSensor cAMP assayMore data for this Ligand-Target Pair
In DepthDetails PubMed