Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50019204
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651113BDBM651113(US20240043470, Compound 1-66)
Affinity DataIC50: 140nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50600763BDBM50600763(CHEMBL5194112 | US20240043470, Compound 1-56)
Affinity DataIC50: 380nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651113BDBM651113(US20240043470, Compound 1-66)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651114BDBM651114(US20240043470, Compound 1-67)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651109BDBM651109(US20240043470, Compound 1-62)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651110BDBM651110(US20240043470, Compound 1-63)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651109BDBM651109(US20240043470, Compound 1-62)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50600762BDBM50600762(CHEMBL5180427 | US20240043470, Compound 1-53)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651110BDBM651110(US20240043470, Compound 1-63)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651114BDBM651114(US20240043470, Compound 1-67)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651130BDBM651130(US20240043470, Compound 1-85)
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651129BDBM651129(US20240043470, Compound 1-84)
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50616641BDBM50616641(CHEMBL5416271)
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651122BDBM651122(US20240043470, Compound 1-77)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651118BDBM651118(US20240043470, Compound 1-73)
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651121BDBM651121(US20240043470, Compound 1-76)
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651129BDBM651129(US20240043470, Compound 1-84)
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651123BDBM651123(US20240043470, Compound 1-78)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651118BDBM651118(US20240043470, Compound 1-73)
Affinity DataIC50: 2.86E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651117BDBM651117(US20240043470, Compound 1-72)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651130BDBM651130(US20240043470, Compound 1-85)
Affinity DataIC50: 3.09E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651125BDBM651125(US20240043470, Compound 1-80)
Affinity DataIC50: 3.13E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651125BDBM651125(US20240043470, Compound 1-80)
Affinity DataIC50: 3.24E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651117BDBM651117(US20240043470, Compound 1-72)
Affinity DataIC50: 3.33E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651120BDBM651120(US20240043470, Compound 1-75)
Affinity DataIC50: 3.35E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50600763BDBM50600763(CHEMBL5194112 | US20240043470, Compound 1-56)
Affinity DataIC50: 3.39E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651122BDBM651122(US20240043470, Compound 1-77)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651124BDBM651124(US20240043470, Compound 1-79)
Affinity DataIC50: 5.98E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50616641BDBM50616641(CHEMBL5416271)
Affinity DataIC50: 8.51E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651120BDBM651120(US20240043470, Compound 1-75)
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651127BDBM651127(US20240043470, Compound 1-82)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651112BDBM651112(US20240043470, Compound 1-65)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651124BDBM651124(US20240043470, Compound 1-79)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651121BDBM651121(US20240043470, Compound 1-76)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50616642BDBM50616642(CHEMBL5421710)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50616643BDBM50616643(CHEMBL5424302)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50616642BDBM50616642(CHEMBL5421710)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50616643BDBM50616643(CHEMBL5424302)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651112BDBM651112(US20240043470, Compound 1-65)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651107BDBM651107(US20240043470, Compound 1-60)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651108BDBM651108(US20240043470, Compound 1-61)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50600762BDBM50600762(CHEMBL5180427 | US20240043470, Compound 1-53)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651106BDBM651106(US20240043470, Compound 1-59)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651105BDBM651105(US20240043470, Compound 1-58)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651106BDBM651106(US20240043470, Compound 1-59)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651105BDBM651105(US20240043470, Compound 1-58)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651123BDBM651123(US20240043470, Compound 1-78)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651107BDBM651107(US20240043470, Compound 1-60)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-5(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651108BDBM651108(US20240043470, Compound 1-61)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5c subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProteasome subunit beta type-8(Human)
Weill Cornell Medicine

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 651119BDBM651119(US20240043470, Compound 1-74)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human 20S immunoproteasome beta-5i subunitMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
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