Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50019820
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Antagonist activity at TRPV4 (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of GSK1016790A induced Ca2+ influx by calcium imag...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Antagonist activity at TRPV4 (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of GSK1016790A induced Ca2+ influx by calcium imag...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 74nMAssay Description:Antagonist activity at TRPV4 (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of GSK1016790A induced Ca2+ influx by calcium imag...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Antagonist activity at TRPV4 (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of GSK1016790A induced Ca2+ influx by calcium imag...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 122nMAssay Description:Antagonist activity at TRPV4 (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of GSK1016790A induced Ca2+ influx by calcium imag...More data for this Ligand-Target Pair
3D Structure (crystal)TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 182nMAssay Description:Antagonist activity at TRPV4 (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of GSK1016790A induced Ca2+ influx by calcium imag...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 203nMAssay Description:Antagonist activity at human TRPV4More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 206nMAssay Description:Antagonist activity at human TRPV4More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 879nMAssay Description:Antagonist activity at TRPV4 (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of GSK1016790A induced Ca2+ influx by calcium imag...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at TRPV4 (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of GSK1016790A induced Ca2+ influx by calcium imag...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at TRPV4 (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of GSK1016790A induced Ca2+ influx by calcium imag...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 4.40E+3nMAssay Description:Antagonist activity at TRPV4 (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of GSK1016790A induced Ca2+ influx by calcium imag...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Beijing Institute of Pharmacology and Toxicology
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Antagonist activity at TRPV4 (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of GSK1016790A induced Ca2+ influx by calcium imag...More data for this Ligand-Target Pair
Ligand InfoSimilars
