Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50019822
Affinity DataIC50: 200nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
3D Structure (crystal)TargetRetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta(Human)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of PDE (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 900nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 6.26E+3nMAssay Description:Mixed type inhibition of human ATX assessed as inhibition constant using LPC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataKi: 6.83E+3nMAssay Description:Mixed type inhibition of human ATX assessed as inhibition constant using LPC as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.21E+4nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 2.12E+4nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 2.21E+4nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 2.44E+4nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 3.73E+4nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 3.84E+4nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 4.08E+4nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 4.18E+4nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 4.66E+4nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 4.83E+4nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 5.37E+4nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 6.30E+4nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetRetinal rod rhodopsin-sensitive cGMP 3',5'-cyclic phosphodiesterase subunit delta(Human)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibition of PDE (unknown origin)More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 7.98E+4nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
TargetEctonucleotide pyrophosphatase/phosphodiesterase family member 2(Mouse)
Bioinnovation Institute
Curated by ChEMBL
Bioinnovation Institute
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of mouse ATX using LPC as substrate preincubated with compound for 15 mins followed by substrate addition measured after 30 mins by Amplex...More data for this Ligand-Target Pair
Ligand InfoSimilars
