Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50019825
TargetReceptor-interacting serine/threonine-protein kinase 2(Human)
The Affiliated Hospital of Qingdao University

Curated by ChEMBL
LigandPNGBDBM50623383(CHEMBL5437324)
Affinity DataIC50: 10nMAssay Description:Inhibition of RIPK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
The Affiliated Hospital of Qingdao University

Curated by ChEMBL
LigandPNGBDBM50623382(CHEMBL5405716)
Affinity DataKd:  490nMAssay Description:Binding affinity to CRBN (unknown origin) assessed as dissociation constant by Tr-FRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetHistone deacetylase 3(Human)
The Affiliated Hospital of Qingdao University

Curated by ChEMBL
LigandPNGBDBM50612668(CHEMBL5282062)
Affinity DataIC50: 560nMAssay Description:Inhibition of His6-tagged Gst fused recombinant human HDAC3 using Ac-Lys-Tyr-Lys(epsilon-acetyl)-AMC as substrate expressed in insect Hi-5 cells meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetHistone deacetylase 1(Human)
The Affiliated Hospital of Qingdao University

Curated by ChEMBL
LigandPNGBDBM50612668(CHEMBL5282062)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of His6-tagged Gst fused recombinant human HDAC1 using Ac-Lys-Tyr-Lys(epsilon-acetyl)-AMC as substrate expressed in insect Hi-5 cells meas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed