Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50020655
Affinity DataIC50: 17nMAssay Description:Inhibition of human EAAT2 transfected in African green monkey COS-1 cells assessed as reduction in [14C]glutamate uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of human EAAT2 transfected in MDCK cells assessed as reduction in [14C]glutamate uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human EAAT1 transfected in African green monkey COS-1 cells assessed as reduction in [14C]glutamate uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of human EAAT3 transfected in MDCK cells assessed as reduction in [14C]glutamate uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 59nMAssay Description:Inhibition of human EAAT2 transfected in African green monkey COS-1 cells assessed as reduction in [14C]glutamate uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 116nMAssay Description:Inhibition of human EAAT1 transfected in African green monkey COS-1 cells assessed as reduction in [14C]glutamate uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human EAAT3 transfected in African green monkey COS-1 cells assessed as reduction in [14C]glutamate uptakeMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human EAAT2 transfected in MDCK cells assessed as reduction in [14C]glutamate uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human EAAT2 transfected in MDCK cells assessed as reduction in L-[3H]glutamate uptake measured upto 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human EAAT3 transfected in African green monkey COS-1 cells assessed as reduction in [14C]glutamate uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human EAAT3 transfected in MDCK cells assessed as reduction in [14C]glutamate uptakeMore data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of human EAAT2 transfected in African green monkey COS-1 cells assessed as reduction in [14C]glutamate uptake incubated for 12 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Inhibition of human EAAT2 transfected in African green monkey COS-1 cells assessed as inhibition of [3H]L-glutamate uptake by measuring inhibition co...More data for this Ligand-Target Pair
Affinity DataKi: 2.30E+4nMAssay Description:Inhibition of human EAAT2 transfected in African green monkey COS-1 cells assessed as inhibition of [3H]L-glutamate uptake by measuring inhibition co...More data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of human EAAT2 transfected in African green monkey COS-1 cells assessed as reduction in [14C]glutamate uptake incubated for 12 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 5.90E+4nMAssay Description:Inhibition of human EAAT2 transfected in African green monkey COS-1 cells assessed as inhibition of [3H]L-glutamate uptake by measuring inhibition co...More data for this Ligand-Target Pair
Affinity DataKi: 6.10E+4nMAssay Description:Inhibition of human EAAT3 transfected in African green monkey COS-1 cells assessed as inhibition of [3H]L-glutamate uptake by measuring inhibition co...More data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of human EAAT1 transfected in African green monkey COS-1 cells assessed as reduction in [14C]glutamate uptake incubated for 12 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: 7.90E+4nMAssay Description:Inhibition of human EAAT1 transfected in African green monkey COS-1 cells assessed as inhibition of [3H]L-glutamate uptake by measuring inhibition co...More data for this Ligand-Target Pair
Affinity DataIC50: 9.60E+4nMAssay Description:Inhibition of human EAAT1 transfected in African green monkey COS-1 cells assessed as reduction in [14C]glutamate uptake incubated for 12 mins by sci...More data for this Ligand-Target Pair
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of human EAAT1 transfected in African green monkey COS-1 cells assessed as inhibition of [3H]L-glutamate uptake by measuring inhibition co...More data for this Ligand-Target Pair
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of human EAAT1 transfected in African green monkey COS-1 cells assessed as inhibition of [3H]L-glutamate uptake by measuring inhibition co...More data for this Ligand-Target Pair
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of human EAAT3 transfected in African green monkey COS-1 cells assessed as inhibition of [3H]L-glutamate uptake by measuring inhibition co...More data for this Ligand-Target Pair
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of human EAAT3 transfected in African green monkey COS-1 cells assessed as inhibition of [3H]L-glutamate uptake by measuring inhibition co...More data for this Ligand-Target Pair
