Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50022265
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650005(CHEMBL5629872)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650004(CHEMBL5631148)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50613442(CHEMBL1233845)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650009(CHEMBL5631045)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650008(CHEMBL5630125)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650007(CHEMBL5630230)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650006(CHEMBL5624765)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650015(CHEMBL5624725)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650014(CHEMBL5624814)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650013(CHEMBL5630899)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650012(CHEMBL5631017)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650013(CHEMBL5630899)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650012(CHEMBL5631017)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650011(CHEMBL5630949)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650010(CHEMBL5630193)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50613442(CHEMBL1233845)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650015(CHEMBL5624725)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650014(CHEMBL5624814)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650007(CHEMBL5630230)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650006(CHEMBL5624765)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650005(CHEMBL5629872)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650004(CHEMBL5631148)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650011(CHEMBL5630949)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650010(CHEMBL5630193)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650009(CHEMBL5631045)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM50650008(CHEMBL5630125)
Affinity DataKi: <0.00500nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM8125(Darunavir (DRV) | CHEMBL1323 | (3R,3aS,6aR)-hexahy...)
Affinity DataKi:  0.0260nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I84V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using a EDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetProtease(Human immunodeficiency virus type 1)TBA
LigandPNGBDBM8125(Darunavir (DRV) | CHEMBL1323 | (3R,3aS,6aR)-hexahy...)
Affinity DataKi:  0.0750nMAssay Description:Binding affinity to drug-resistant HIV-1 protease I50V/A71V mutant expressed in Escherichia coli TAP-106 cells assessed as inhibition constant using ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed