Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50019302
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617852BDBM50617852(CHEMBL5400665)
Affinity DataIC50: 21nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617857BDBM50617857(CHEMBL5409784)
Affinity DataIC50: 57nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617845BDBM50617845(CHEMBL5423121)
Affinity DataIC50: 72nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617843BDBM50617843(CHEMBL5403672)
Affinity DataIC50: 90nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617847BDBM50617847(CHEMBL5406504)
Affinity DataIC50: 90nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617851BDBM50617851(CHEMBL5420904)
Affinity DataIC50: 100nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617852BDBM50617852(CHEMBL5400665)
Affinity DataIC50: 100nMAssay Description:Inhibition of Escherichia coli DNA gyrase supercoiling activity using relaxed pBR322 DNA as substrate preincubated for 5 mins followed by enzyme addi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617854BDBM50617854(CHEMBL5422268)
Affinity DataIC50: 120nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617848BDBM50617848(CHEMBL5424692)
Affinity DataIC50: 120nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617856BDBM50617856(CHEMBL5435353)
Affinity DataIC50: 160nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617842BDBM50617842(CHEMBL5404831)
Affinity DataIC50: 160nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617850BDBM50617850(CHEMBL5410417)
Affinity DataIC50: 180nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617858BDBM50617858(CHEMBL5424981)
Affinity DataIC50: 190nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617849BDBM50617849(CHEMBL5405573)
Affinity DataIC50: 230nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617855BDBM50617855(CHEMBL5430363)
Affinity DataIC50: 250nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617853BDBM50617853(CHEMBL5409273)
Affinity DataIC50: 270nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617844BDBM50617844(CHEMBL5395093)
Affinity DataIC50: 290nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617846BDBM50617846(CHEMBL5422850)
Affinity DataIC50: 580nMAssay Description:Inhibition of Escherichia coli DNA gyrase ATPase activity incubated for 80 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617852BDBM50617852(CHEMBL5400665)
Affinity DataIC50: 900nMAssay Description:Inhibition of human ERG expressed in CHO cells by automated path clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetDNA topoisomerase 2-alpha(Human)
Roche Pharma Research & Early Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50617852BDBM50617852(CHEMBL5400665)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human topoisomerase 2 alpha decatenation activity using kDNA as substrate preincubated for 5 mins followed by enzyme addition and measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed