Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50019431
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 60nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 100nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human A498 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 180nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human A498 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 190nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 210nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 230nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human A498 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 280nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human A498 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 290nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human A498 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 290nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human WPMY-1 cells assessed as transcriptional activation incubated for 72 hrs under normoxic condition ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 310nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human A498 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 320nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 360nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human A498 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 380nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human WPMY-1 cells assessed as transcriptional activation incubated for 72 hrs under normoxic condition ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 430nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human WPMY-1 cells assessed as transcriptional activation incubated for 72 hrs under normoxic condition ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 440nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human A498 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 450nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human WPMY-1 cells assessed as transcriptional activation incubated for 72 hrs under normoxic condition ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 470nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human A498 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 580nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human A498 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 580nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human WPMY-1 cells assessed as transcriptional activation incubated for 72 hrs under normoxic condition ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 580nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human A498 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 600nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human WPMY-1 cells assessed as transcriptional activation incubated for 72 hrs under normoxic condition ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 630nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human DU-145 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition b...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 630nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human A498 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition by ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 670nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human WPMY-1 cells assessed as transcriptional activation incubated for 72 hrs under normoxic condition ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 680nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human WPMY-1 cells assessed as transcriptional activation incubated for 72 hrs under normoxic condition ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 730nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human WPMY-1 cells assessed as transcriptional activation incubated for 72 hrs under normoxic condition ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 770nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human DU-145 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition b...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 780nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human WPMY-1 cells assessed as transcriptional activation incubated for 72 hrs under normoxic condition ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 830nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human DU-145 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition b...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 840nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human WPMY-1 cells assessed as transcriptional activation incubated for 72 hrs under normoxic condition ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 860nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human DU-145 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition b...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 910nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human WPMY-1 cells assessed as transcriptional activation incubated for 72 hrs under normoxic condition ...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 1.17E+3nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 1.19E+3nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human DU-145 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition b...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 1.26E+3nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human DU-145 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition b...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 1.29E+3nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human DU-145 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition b...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 1.38E+3nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human DU-145 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition b...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 1.50E+3nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human DU-145 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition b...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 1.62E+3nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human DU-145 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition b...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 1.72E+3nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human DU-145 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition b...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 1.76E+3nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human RPTEC assessed as transcriptional activation incubated for 72 hrs under normoxic condition by luci...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Human)
Universidad Complutense of Madrid
Curated by ChEMBL
Universidad Complutense of Madrid
Curated by ChEMBL
Affinity DataEC50: 1.77E+3nMAssay Description:Agonist activity at GAL4-tagged PPARalpha in human DU-145 cells assessed as transcriptional activation incubated for 72 hrs under hypoxic condition b...More data for this Ligand-Target Pair













