Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50019420
TargetProtein arginine N-methyltransferase 1(Human)
Minzu University of China

Curated by ChEMBL
LigandPNGBDBM50388602(FURAMIDINE)
Affinity DataIC50: 310nMAssay Description:Displacement of [3H]SAM from PRMT1 (unknown origin) preincubated for 15 mins followed by [3H]SAM addition measured after 60 mins by radiometric/lumin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Minzu University of China

Curated by ChEMBL
LigandPNGBDBM50619070(CHEMBL5428645)
Affinity DataIC50: 7.07E+3nMAssay Description:Displacement of [3H]SAM from PRMT1 (unknown origin) preincubated for 15 mins followed by [3H]SAM addition measured after 60 mins by radiometric/lumin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 1(Human)
Minzu University of China

Curated by ChEMBL
LigandPNGBDBM50619069(CHEMBL5403175)
Affinity DataIC50: 1.18E+4nMAssay Description:Displacement of [3H]SAM from PRMT1 (unknown origin) preincubated for 15 mins followed by [3H]SAM addition measured after 60 mins by radiometric/lumin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed