Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50020991
LigandPNGBDBM50575072(Fisogatinib | BLU-111362 | BLU-554 | BLU111362 | X...)
Affinity DataIC50: 3nMAssay Description:Inhibition of FGFR4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50233461(CHEMBL4068896)
Affinity DataIC50: 3nMAssay Description:Inhibition of C-terminal Histidine-tagged human FGFR4 (570 to 578 residues) expressed in Sf21 insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50635830(CHEMBL5517830)
Affinity DataIC50: 48nMAssay Description:Inhibition of N-terminal 6xHis-tagged human FGFR4 (445 to 753 residues) transfected in Escherichia coli Rossetta cells incubated for 30 mins by ADP-G...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50635831(CHEMBL5542790)
Affinity DataIC50: 75nMAssay Description:Inhibition of human FGFR4 using poly (Glu, Tyr)4:1 as substrate measured after 30 mins by ADP-Glo reagent based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50575072(Fisogatinib | BLU-111362 | BLU-554 | BLU111362 | X...)
Affinity DataIC50: 150nMAssay Description:Inhibition of FGFR3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50233461(CHEMBL4068896)
Affinity DataIC50: 150nMAssay Description:Inhibition of FGFR3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50635830(CHEMBL5517830)
Affinity DataIC50: 193nMAssay Description:Inhibition of FGFR4 C477A mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50575072(Fisogatinib | BLU-111362 | BLU-554 | BLU111362 | X...)
Affinity DataIC50: 493nMAssay Description:Inhibition of FGFR2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50233461(CHEMBL4068896)
Affinity DataIC50: 493nMAssay Description:Inhibition of FGFR2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50575072(Fisogatinib | BLU-111362 | BLU-554 | BLU111362 | X...)
Affinity DataIC50: 591nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50233461(CHEMBL4068896)
Affinity DataIC50: 591nMAssay Description:Inhibition of FGFR1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50635830(CHEMBL5517830)
Affinity DataIC50: 602nMAssay Description:Inhibition of FGFR4 C552A mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50635830(CHEMBL5517830)
Affinity DataIC50: 977nMAssay Description:Inhibition of N-terminal 6xHis-tagged human FGFR3 (450 to 758 residues) transfected in Escherichia coli Rossetta cells incubated for 30 mins by ADP-G...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50635830(CHEMBL5517830)
Affinity DataIC50: 1.53E+3nMAssay Description:Inhibition of FGFR4 C552A/C477A double mutant (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50635830(CHEMBL5517830)
Affinity DataIC50: 2.41E+3nMAssay Description:Inhibition of N-terminal 6xHis-tagged human FGFR2 (453 to 770 residues) transfected in Escherichia coli Rossetta cells incubated for 30 mins by ADP-G...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50635830(CHEMBL5517830)
Affinity DataIC50: 2.58E+3nMAssay Description:Inhibition of N-terminal 6xHis-tagged human FGFR1 (456 to 765 residues) transfected in Escherichia coli Rossetta cells incubated for 30 mins by ADP-G...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50635831(CHEMBL5542790)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of FGFR3 (unknown origin) incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50635831(CHEMBL5542790)
Affinity DataIC50: 3.55E+4nMAssay Description:Inhibition of FGFR2 (unknown origin) incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50635831(CHEMBL5542790)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of FGFR1 (unknown origin) incubated for 30 mins by ADP-Glo assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed