Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50021420
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640499(CHEMBL5573022)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of N-terminal GST-tagged recombinant full length human c-Src kinase expressed in baculovirus-infected Sf9 cells preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640510(CHEMBL5572163)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of N-terminal GST-tagged recombinant full length human c-Src kinase expressed in baculovirus-infected Sf9 cells preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 61nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640494(CHEMBL5593071)
Affinity DataIC50: 76nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640511(CHEMBL5591671)
Affinity DataIC50: 98nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640495(CHEMBL5569888)
Affinity DataIC50: 98nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640498(CHEMBL5568829)
Affinity DataIC50: 105nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640510(CHEMBL5572163)
Affinity DataIC50: 122nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human BRD4 BD1 expressed in Escherichia coli incubated for 15 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640510(CHEMBL5572163)
Affinity DataIC50: 133nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640506(CHEMBL5572942)
Affinity DataIC50: 185nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640509(CHEMBL5574101)
Affinity DataIC50: 202nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640496(CHEMBL5537100)
Affinity DataIC50: 219nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640504(CHEMBL5573987)
Affinity DataIC50: 219nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640499(CHEMBL5573022)
Affinity DataIC50: 235nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640501(CHEMBL5591616)
Affinity DataIC50: 279nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640503(CHEMBL5569521)
Affinity DataIC50: 305nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640493(CHEMBL5572493)
Affinity DataIC50: 445nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640507(CHEMBL5570665)
Affinity DataIC50: 547nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640500(CHEMBL5575293)
Affinity DataIC50: 547nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640508(CHEMBL5573535)
Affinity DataIC50: 799nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640497(CHEMBL5556700)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640505(CHEMBL5570956)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Shenzhen University

Curated by ChEMBL
LigandPNGBDBM50640502(CHEMBL5568695)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of His6-tagged recombinant BRD4 BD1 domain (44 to 168 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) incubated for 0.5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed