Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50020581
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631541(CHEMBL5412813)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631547(CHEMBL5418460)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631548(CHEMBL5418271)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631545(CHEMBL5414839)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50520131(CHEMBL4588661)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631546(CHEMBL5411289)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631549(CHEMBL5432148)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631550(CHEMBL5421916)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631539(CHEMBL5417425)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631540(CHEMBL5422217)
Affinity DataKi:  0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50605355(CHEMBL5170717)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631538(CHEMBL5409903)
Affinity DataKi: <0.0200nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631535(CHEMBL5398730)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631534(CHEMBL5398302)
Affinity DataKi:  0.0260nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631544(CHEMBL5405792)
Affinity DataKi:  0.0270nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631542(CHEMBL5401138)
Affinity DataKi:  0.0330nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631531(CHEMBL5431390)
Affinity DataKi:  0.0370nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631543(CHEMBL5440128)
Affinity DataKi:  0.0390nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631537(CHEMBL5425914)
Affinity DataKi:  0.0470nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50520130(CHEMBL4435250)
Affinity DataKi:  0.0490nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631532(CHEMBL5401714)
Affinity DataKi:  0.0510nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631533(CHEMBL5434280)
Affinity DataKi:  0.0790nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631536(CHEMBL5404726)
Affinity DataKi:  0.100nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631530(CHEMBL5440410)
Affinity DataKi:  0.570nMAssay Description:Inhibition of 6His-SUMO tagged human WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold (DE3) cells incubated for 1 hr by TR-FRET assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50631529(CHEMBL5415680)
Affinity DataEC50:  4nMAssay Description:Induction of WDR5 degradation in human MV4-11 cells incubated for 18 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetWD repeat-containing protein 5(Human)
Institute of Chemical Biology

Curated by ChEMBL
LigandPNGBDBM50164794(CHEMBL3798846 | US11174250, Example Table4.1.1 | U...)
Affinity DataKi:  30nMAssay Description:Binding affinity to WDR5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed