Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50020589
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631628(CHEMBL5399086)
Affinity DataIC50: 8.40nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631627(CHEMBL5422157)
Affinity DataIC50: 8.90nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631636(CHEMBL5421315)
Affinity DataIC50: 10nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631626(CHEMBL5394571)
Affinity DataIC50: 11nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631628(CHEMBL5399086)
Affinity DataIC50: 12nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631627(CHEMBL5422157)
Affinity DataIC50: 15nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631625(CHEMBL5422650)
Affinity DataIC50: 15nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631623(CHEMBL5439152)
Affinity DataIC50: 17nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631624(CHEMBL5405846)
Affinity DataIC50: 18nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631629(CHEMBL5420072)
Affinity DataIC50: 18nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631633(CHEMBL5395213)
Affinity DataIC50: 19nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631635(CHEMBL5432640)
Affinity DataIC50: 21nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631632(CHEMBL5398776)
Affinity DataIC50: 21nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631631(CHEMBL5431364)
Affinity DataIC50: 25nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631631(CHEMBL5431364)
Affinity DataIC50: 25nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631630(CHEMBL5405431)
Affinity DataIC50: 26nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631634(CHEMBL5415959)
Affinity DataIC50: 28nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631632(CHEMBL5398776)
Affinity DataIC50: 31nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631633(CHEMBL5395213)
Affinity DataIC50: 32nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631630(CHEMBL5405431)
Affinity DataIC50: 54nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631629(CHEMBL5420072)
Affinity DataIC50: 55nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631634(CHEMBL5415959)
Affinity DataIC50: 77nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631626(CHEMBL5394571)
Affinity DataIC50: 137nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631636(CHEMBL5421315)
Affinity DataIC50: 169nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631622(CHEMBL5394825)
Affinity DataIC50: 216nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in digitonin-permeabilized HEK293 cells incubated for 10 mins by NanoBRET target e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631635(CHEMBL5432640)
Affinity DataIC50: 287nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631625(CHEMBL5422650)
Affinity DataIC50: 292nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631622(CHEMBL5394825)
Affinity DataIC50: 302nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631623(CHEMBL5439152)
Affinity DataIC50: 388nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed
TargetProtein cereblon(Human)
Boehringer Ingelheim Rcv

Curated by ChEMBL
LigandPNGBDBM50631624(CHEMBL5405846)
Affinity DataIC50: 622nMAssay Description:Binding affinity to Nano-Luc fused CRBN (unknown origin) expressed in live HEK293 cells incubated for 30 mins by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2024
Entry Details
PubMed