Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50021517
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641425BDBM50641425(CHEMBL5563688)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641423BDBM50641423(CHEMBL5566630)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641424BDBM50641424(CHEMBL5591635)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641419BDBM50641419(CHEMBL5595209)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641410BDBM50641410(CHEMBL5579677)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641429BDBM50641429(CHEMBL5571078)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641421BDBM50641421(CHEMBL5565603)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641422BDBM50641422(CHEMBL5579700)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641420BDBM50641420(CHEMBL5572811)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641437BDBM50641437(CHEMBL5563776)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641417BDBM50641417(CHEMBL5569108)
Affinity DataIC50: 1nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641432BDBM50641432(CHEMBL5563712)
Affinity DataIC50: 1nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641438BDBM50641438(CHEMBL5572936)
Affinity DataIC50: 1nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 413450BDBM413450(US10407446, Example 3 | 7-methyl-2-((7-methyl-[1,2...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641436BDBM50641436(CHEMBL5575123)
Affinity DataIC50: 1nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641408BDBM50641408(CHEMBL5572260)
Affinity DataIC50: 1nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641439BDBM50641439(CHEMBL5570412)
Affinity DataIC50: 1nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641441BDBM50641441(CHEMBL5592744)
Affinity DataIC50: 2nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641430BDBM50641430(CHEMBL5566668)
Affinity DataIC50: 2nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641416BDBM50641416(CHEMBL5571138)
Affinity DataIC50: 3nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641440BDBM50641440(CHEMBL5571620)
Affinity DataIC50: 3nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641428BDBM50641428(CHEMBL5591387)
Affinity DataIC50: 4nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641442BDBM50641442(CHEMBL5565467)
Affinity DataIC50: 5nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641409BDBM50641409(CHEMBL5574317)
Affinity DataIC50: 5nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641414BDBM50641414(CHEMBL5564989)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641418BDBM50641418(CHEMBL5592925)
Affinity DataIC50: 6nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641434BDBM50641434(CHEMBL5572732)
Affinity DataIC50: 6nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641406BDBM50641406(CHEMBL5572444)
Affinity DataIC50: 6nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641427BDBM50641427(CHEMBL5569624)
Affinity DataIC50: 6nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641433BDBM50641433(CHEMBL5595206)
Affinity DataIC50: 8nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641426BDBM50641426(CHEMBL5567517)
Affinity DataIC50: 8nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641435BDBM50641435(CHEMBL5572075)
Affinity DataIC50: 9nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641413BDBM50641413(CHEMBL5564999)
Affinity DataIC50: 9.60nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641431BDBM50641431(CHEMBL5571804)
Affinity DataIC50: 10nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641443BDBM50641443(CHEMBL5563030)
Affinity DataIC50: 12nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641407BDBM50641407(CHEMBL5571528)
Affinity DataIC50: 13nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641412BDBM50641412(CHEMBL5595128)
Affinity DataIC50: 13nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641411BDBM50641411(CHEMBL5595223)
Affinity DataIC50: 25nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetDNA-dependent protein kinase catalytic subunit(Human)
West China Hospital

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50641415BDBM50641415(CHEMBL5575061)
Affinity DataIC50: 161nMAssay Description:Inhibition of human DNA-PK incubated for 30 mins in presence of Mg/ATP by HTRF methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed