Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50019765
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50622896(CHEMBL5415555)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to GLUT1 (unknown origin) assessed as dissociation constant at 800 uM by MST assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50622897(CHEMBL3895916)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to GLUT1 (unknown origin) assessed as dissociation constant at 800 uM by MST assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50622895(CHEMBL5396476)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to GLUT1 (unknown origin) assessed as dissociation constant at 800 uM by MST assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50622895(CHEMBL5396476)
Affinity DataIC50: 3.46E+3nMAssay Description:Inhibition of GLUT1 in human MCF7 cells assessed as ATP production incubated for 24 hrs in presence of 0.1 mM glucoseMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50622895(CHEMBL5396476)
Affinity DataIC50: 1.80E+5nMAssay Description:Inhibition of GLUT1 in human MCF7 cells assessed as ATP production incubated for 24 hrs in presence of 10 mM glucoseMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed