Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50021519
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641492(CHEMBL5569161)
Affinity DataIC50: 111nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641496(CHEMBL5568622)
Affinity DataIC50: 135nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641476(CHEMBL5567043)
Affinity DataIC50: 136nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641488(CHEMBL5563043)
Affinity DataIC50: 155nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641501(CHEMBL5590984)
Affinity DataIC50: 164nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataIC50: 186nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641486(CHEMBL5569094)
Affinity DataIC50: 196nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641475(CHEMBL5555360)
Affinity DataIC50: 200nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641463(CHEMBL5565769)
Affinity DataIC50: 212nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641503(CHEMBL5565943)
Affinity DataIC50: 214nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641474(CHEMBL5575877)
Affinity DataIC50: 250nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641473(CHEMBL5593403)
Affinity DataIC50: 295nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641465(CHEMBL5593664)
Affinity DataIC50: 332nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641494(CHEMBL5563792)
Affinity DataIC50: 443nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641498(CHEMBL5570562)
Affinity DataIC50: 452nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641502(CHEMBL5594723)
Affinity DataIC50: 461nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641467(CHEMBL5573730)
Affinity DataIC50: 505nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641485(CHEMBL5571572)
Affinity DataIC50: 544nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641495(CHEMBL5573769)
Affinity DataIC50: 597nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641487(CHEMBL5571059)
Affinity DataIC50: 625nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641470(CHEMBL5571115)
Affinity DataIC50: 655nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641489(CHEMBL5574997)
Affinity DataIC50: 716nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641496(CHEMBL5568622)
Affinity DataKi:  780nMAssay Description:Displacement of fluormone AL green from AR-LBD (unknown origin) incubated for 3 hrs by PolarScreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641472(CHEMBL5563225)
Affinity DataIC50: 792nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641466(CHEMBL5589667)
Affinity DataIC50: 806nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641456(CHEMBL5574098)
Affinity DataIC50: 831nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641457(CHEMBL5594380)
Affinity DataIC50: 999nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641469(CHEMBL5563558)
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641497(CHEMBL5574051)
Affinity DataIC50: 1.06E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641483(CHEMBL5572979)
Affinity DataIC50: 1.08E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641458(CHEMBL5572389)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641460(CHEMBL5584051)
Affinity DataIC50: 1.13E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641468(CHEMBL5569474)
Affinity DataIC50: 1.14E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641493(CHEMBL5565870)
Affinity DataIC50: 1.15E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641481(CHEMBL5571579)
Affinity DataIC50: 1.23E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641491(CHEMBL5572527)
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641462(CHEMBL5572462)
Affinity DataIC50: 1.32E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641464(CHEMBL5574403)
Affinity DataIC50: 1.42E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641499(CHEMBL5573540)
Affinity DataIC50: 1.54E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641471(CHEMBL5566095)
Affinity DataIC50: 1.58E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641490(CHEMBL5564844)
Affinity DataIC50: 1.59E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641461(CHEMBL5571658)
Affinity DataIC50: 1.63E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641484(CHEMBL5564208)
Affinity DataIC50: 1.64E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641455(CHEMBL5572524)
Affinity DataIC50: 1.76E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50425732(Xtandi | ENZALUTAMIDE | US10053433, FC 4.129 | US1...)
Affinity DataKi:  2.37E+3nMAssay Description:Displacement of fluormone AL green from AR-LBD (unknown origin) incubated for 3 hrs by PolarScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641480(CHEMBL5574257)
Affinity DataIC50: 2.58E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641500(CHEMBL5590394)
Affinity DataIC50: 2.61E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641477(CHEMBL5574975)
Affinity DataIC50: 3.14E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein cereblon/CUL4A/AR(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641478(CHEMBL5565106)
Affinity DataIC50: 3.38E+3nMAssay Description:Antagonist activity at AR in human LNCaP cells assessed as reduction in R1881-induced AR transcriptional activity preincubated for 60 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProgesterone receptor(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50641496(CHEMBL5568622)
Affinity DataIC50: 3.50E+3nMAssay Description:Antagonist activity at PR in HEK293T cells assessed as reduction in transcriptional activity incubated for 24 hrs by britelite plus reagent based pla...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
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