Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50021677
Affinity DataKd: 5.5nMAssay Description:Binding affinity to human BRD3 assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKd: 5.60nMAssay Description:Binding affinity to human BRD2 assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKd: 6.70nMAssay Description:Binding affinity to human BRD4 BD1 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding affinity to human BRD4 BD2 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Binding affinity to human BRD4 BD2 expressed in Escherichia coli BL21 (DE3) by TR-FRET analysisMore data for this Ligand-Target Pair
Affinity DataKd: 14nMAssay Description:Binding affinity to human BRDT assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of human BRD4 BD2 (44 to 460 residues) by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of human BRD4 BD1 (44 to 460 residues) by Alphascreen assayMore data for this Ligand-Target Pair
Affinity DataKd: 29nMAssay Description:Binding affinity to human BRD4 BD1 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: 32nMAssay Description:Binding affinity to human BRD4 BD1 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Binding affinity to human BRD4 BD1 expressed in Escherichia coli BL21 (DE3) by TR-FRET analysisMore data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Binding affinity to human BRD4 BD1 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: 37nMAssay Description:Binding affinity to human BRD4 BD1 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: 40nMAssay Description:Binding affinity to human BRD4 BD1 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 86nMAssay Description:Inhibition of human BRD3More data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding affinity to human BRD4 BD2 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 144nMAssay Description:Inhibition of human BRDTMore data for this Ligand-Target Pair
Affinity DataIC50: 163nMAssay Description:Inhibition of human BRD2More data for this Ligand-Target Pair
Affinity DataKd: 180nMAssay Description:Binding affinity to human BRD4 BD2 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: 190nMAssay Description:Binding affinity to human BRD4 BD2 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: 220nMAssay Description:Binding affinity to human BRD4 BD2 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: 260nMAssay Description:Binding affinity to human BRD4 BD1 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: 293nMAssay Description:Binding affinity to human BRD4 BD2 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKd: 510nMAssay Description:Binding affinity to human BRD4 BD1 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: 630nMAssay Description:Binding affinity to human BRD4 BD2 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: 900nMAssay Description:Binding affinity to human BRD4 BD2 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Binding affinity to human BRD4 BD1 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: 2.20E+3nMAssay Description:Binding affinity to human BRD4 BD2 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: >5.00E+3nMAssay Description:Binding affinity to human BRD4 BD1 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: >5.00E+3nMAssay Description:Binding affinity to human BRD4 BD2 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: >5.00E+3nMAssay Description:Binding affinity to human BRD4 BD1 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
Affinity DataKd: >5.00E+3nMAssay Description:Binding affinity to human BRD4 BD2 expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant by bromodomain analysisMore data for this Ligand-Target Pair
