Compile Data Set for Download or QSAR
Report error Found 65 Enz. Inhib. hit(s) with all data for entry = 50021431
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50006932(CHEMBL3237245)
Affinity DataKi:  1nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640677(CHEMBL5571025)
Affinity DataKi:  1.90nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640670(CHEMBL5595521)
Affinity DataKi:  6.40nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640677(CHEMBL5571025)
Affinity DataKi:  7.60nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640676(CHEMBL5570595)
Affinity DataKi:  9.10nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640672(CHEMBL5567314)
Affinity DataKi:  12nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50006932(CHEMBL3237245)
Affinity DataKi:  12nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640677(CHEMBL5571025)
Affinity DataIC50: 19nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640676(CHEMBL5570595)
Affinity DataIC50: 22nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640670(CHEMBL5595521)
Affinity DataKi:  24nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50006932(CHEMBL3237245)
Affinity DataIC50: 29nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640667(CHEMBL5567570)
Affinity DataKi:  30nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640671(CHEMBL5572451)
Affinity DataKi:  31nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640672(CHEMBL5567314)
Affinity DataKi:  32nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640678(CHEMBL5556087)
Affinity DataKi:  41nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640657(CHEMBL5569386)
Affinity DataKi:  51nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640670(CHEMBL5595521)
Affinity DataIC50: 54nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50006932(CHEMBL3237245)
Affinity DataIC50: 63nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640662(CHEMBL5555837)
Affinity DataKi:  66nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640673(CHEMBL5573249)
Affinity DataKi:  68nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640668(CHEMBL5590315)
Affinity DataKi:  68nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640676(CHEMBL5570595)
Affinity DataIC50: 69nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640672(CHEMBL5567314)
Affinity DataIC50: 72nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640655(CHEMBL5573658)
Affinity DataKi:  74nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50593809(CHEMBL5181633)
Affinity DataKi:  76nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640658(CHEMBL5564155)
Affinity DataKi:  78nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640656(CHEMBL5574547)
Affinity DataKi:  82nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640677(CHEMBL5571025)
Affinity DataIC50: 89nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640678(CHEMBL5556087)
Affinity DataIC50: 92nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640675(CHEMBL5593633)
Affinity DataKi:  100nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640660(CHEMBL5590204)
Affinity DataKi:  106nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640670(CHEMBL5595521)
Affinity DataIC50: 111nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640669(CHEMBL5557583)
Affinity DataKi:  116nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640672(CHEMBL5567314)
Affinity DataIC50: 136nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640659(CHEMBL5571910)
Affinity DataKi:  141nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50593788(CHEMBL5172581)
Affinity DataKi:  146nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640667(CHEMBL5567570)
Affinity DataIC50: 226nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640671(CHEMBL5572451)
Affinity DataIC50: 228nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640666(CHEMBL5563080)
Affinity DataKi:  316nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640657(CHEMBL5569386)
Affinity DataIC50: 325nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640674(CHEMBL5594768)
Affinity DataKi:  351nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640654(CHEMBL5583856)
Affinity DataKi:  351nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640662(CHEMBL5555837)
Affinity DataIC50: 399nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640668(CHEMBL5590315)
Affinity DataIC50: 407nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640673(CHEMBL5573249)
Affinity DataIC50: 408nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640655(CHEMBL5573658)
Affinity DataIC50: 439nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50593809(CHEMBL5181633)
Affinity DataIC50: 449nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640664(CHEMBL5543048)
Affinity DataKi:  452nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) assessed as inhibition constant by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640658(CHEMBL5564155)
Affinity DataIC50: 458nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
The State University of New Jersey

Curated by ChEMBL
LigandPNGBDBM50640656(CHEMBL5574547)
Affinity DataIC50: 476nMAssay Description:Inhibition of Keap1-Nrf2 protein-protein interaction (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
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