Compile Data Set for Download or QSAR
Report error Found 82 Enz. Inhib. hit(s) with all data for entry = 50021678
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of c-MET (unknown origin) phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM180270(US9133162, Example 1)
Affinity DataIC50: 1nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643349(CHEMBL5565630)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50021574(CHEBI:72317 | CABOZANTINIB | BMS-907351 | Cometriq...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of c-MET (unknown origin) phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643352(CHEMBL5570772)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643350(CHEMBL5594055)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM28031(N-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorop...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50172078(LY-2801653 | Merestinib | US11952364, Example Mere...)
Affinity DataIC50: 2nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50172078(LY-2801653 | Merestinib | US11952364, Example Mere...)
Affinity DataKi:  2nMAssay Description:Inhibition of c-MET (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643347(CHEMBL5572673)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643339(CHEMBL5569554)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643332(CHEMBL5574768)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM387260(US9938274, Comparative Compound B)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643334(CHEMBL5575269)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643333(CHEMBL5563765)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM180270(US9133162, Example 1)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of c-MET (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM336532(US9745283, Example 5)
Affinity DataIC50: 7nMAssay Description:Inhibition of AXL (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50021574(CHEBI:72317 | CABOZANTINIB | BMS-907351 | Cometriq...)
Affinity DataIC50: 7nMAssay Description:Inhibition of AXL (unknown origin) phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643345(CHEMBL5574080)
Affinity DataIC50: 7.40nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM28031(N-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorop...)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of recombinant MET (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)
Affinity DataIC50: 11nMAssay Description:Inhibition of AXL (unknown origin) phosphorylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM336532(US9745283, Example 5)
Affinity DataIC50: 12nMAssay Description:Inhibition of c-MET (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643336(CHEMBL5575968)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643341(CHEMBL5569183)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643345(CHEMBL5574080)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643346(CHEMBL5574121)
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643337(CHEMBL5570992)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643343(CHEMBL5595612)
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643335(CHEMBL5572537)
Affinity DataIC50: 24nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643338(CHEMBL5569411)
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643344(CHEMBL5571226)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643332(CHEMBL5574768)
Affinity DataIC50: 28nMAssay Description:Inhibition of recombinant MET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643340(CHEMBL5572307)
Affinity DataIC50: 28nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643331(CHEMBL5573302)
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643352(CHEMBL5570772)
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant MET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643342(CHEMBL5574134)
Affinity DataIC50: 34nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643332(CHEMBL5574768)
Affinity DataIC50: 34nMAssay Description:Inhibition of recombinant VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643337(CHEMBL5570992)
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant MET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643350(CHEMBL5594055)
Affinity DataIC50: 47nMAssay Description:Inhibition of recombinant MET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643333(CHEMBL5563765)
Affinity DataIC50: 47nMAssay Description:Inhibition of recombinant MET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643331(CHEMBL5573302)
Affinity DataIC50: 49nMAssay Description:Inhibition of recombinant VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643331(CHEMBL5573302)
Affinity DataIC50: 51nMAssay Description:Inhibition of recombinant MET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643339(CHEMBL5569554)
Affinity DataIC50: 55nMAssay Description:Inhibition of recombinant MET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643348(CHEMBL5570274)
Affinity DataIC50: 57nMAssay Description:Inhibition of recombinant MET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643334(CHEMBL5575269)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant MET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643336(CHEMBL5575968)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643333(CHEMBL5563765)
Affinity DataIC50: 62nMAssay Description:Inhibition of recombinant VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643337(CHEMBL5570992)
Affinity DataIC50: 63nMAssay Description:Inhibition of recombinant VEGFR-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643335(CHEMBL5572537)
Affinity DataIC50: 68nMAssay Description:Inhibition of recombinant MET (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50643351(CHEMBL5595200)
Affinity DataIC50: 69nMAssay Description:Inhibition of recombinant AXL (unknown origin) by FRET based Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
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