Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50021679
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM28661(GW501516 | CHEMBL38943 | 2-{2-methyl-4-[({4-methyl...)
Affinity DataEC50:  4nMAssay Description:Agonist activity at GAL4-tagged human PPARbeta/delta transfected in african green monkey COS7 cells assessed transcriptional activation incubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50030474(US9562012, rosiglitazone | CHEBI:50122 | Avandamet...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human PPARgamma transfected in african green monkey COS7 cells assessed transcriptional activation incubated for 24 hrs by lucife...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50643354(CHEMBL5589777)
Affinity DataEC50:  226nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha transfected in african green monkey COS7 cells assessed transcriptional activation incubated for 24 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50643353(CHEMBL5574026)
Affinity DataEC50:  493nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha transfected in african green monkey COS7 cells assessed transcriptional activation incubated for 24 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50643355(CHEMBL5566513)
Affinity DataEC50:  1.48E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARbeta/delta transfected in african green monkey COS7 cells assessed transcriptional activation incubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50643355(CHEMBL5566513)
Affinity DataEC50:  3.26E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha transfected in african green monkey COS7 cells assessed transcriptional activation incubated for 24 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50643353(CHEMBL5574026)
Affinity DataEC50:  3.27E+3nMAssay Description:Agonist activity at human PPARgamma transfected in african green monkey COS7 cells assessed transcriptional activation incubated for 24 hrs by lucife...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM24566(JMC515449 Compound 1 | Wyeth 14,643 | 2-({4-chloro...)
Affinity DataEC50:  4.19E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha transfected in african green monkey COS7 cells assessed transcriptional activation incubated for 24 h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Valencia

Curated by ChEMBL
LigandPNGBDBM50643354(CHEMBL5589777)
Affinity DataEC50:  5.54E+3nMAssay Description:Agonist activity at human PPARgamma transfected in african green monkey COS7 cells assessed transcriptional activation incubated for 24 hrs by lucife...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed