Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50021620
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM624800(US11780854, Example 48)
Affinity DataIC50: 1nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642776(CHEMBL5572635)
Affinity DataIC50: 1nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642762(CHEMBL5564592)
Affinity DataIC50: 2nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642775(CHEMBL5574218)
Affinity DataIC50: 2nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642772(CHEMBL5565890)
Affinity DataIC50: 2nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642773(CHEMBL5563061)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642774(CHEMBL5572587)
Affinity DataIC50: 3nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642771(CHEMBL5572628)
Affinity DataIC50: 4nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642770(CHEMBL5594033)
Affinity DataIC50: 4nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642759(CHEMBL5575448)
Affinity DataIC50: 4nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642761(CHEMBL5567289)
Affinity DataIC50: 9nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50431015(CHEMBL2338329 | US9115085, Compound A Form A | US9...)
Affinity DataIC50: 14nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642760(CHEMBL5571964)
Affinity DataIC50: 19nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642767(CHEMBL5562929)
Affinity DataIC50: 37nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642763(CHEMBL5583677)
Affinity DataIC50: 87nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642769(CHEMBL5594247)
Affinity DataIC50: 291nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642768(CHEMBL5572863)
Affinity DataIC50: 297nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642764(CHEMBL5572667)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetGlucocorticoid receptor(Human)TBA
LigandPNGBDBM50642773(CHEMBL5563061)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of glucocorticoid receptor (unknown origin) by KINOMEscan analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50642773(CHEMBL5563061)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of androgen receptor (unknown origin) by KINOMEscan analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642766(CHEMBL5572357)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetEgl nine homolog 1(Human)TBA
LigandPNGBDBM50642765(CHEMBL5570245)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of PHD2 (unknown origin) preincubated for 30 mins followed by substrate addition and measured after 30 mins by HTS plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed