Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50020068
TargetBromodomain-containing protein 4(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 49nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 53nMAssay Description:Inhibition of BRD4 (unknown origin) by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 103nMAssay Description:Binding affinity to BRDT bromodomain (unknown origin) by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 124nMAssay Description:Binding affinity to BRDT bromodomain (unknown origin) by alpha screen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  188nMAssay Description:Binding affinity to his tagged BRDT bromodomain (unknown origin) assessed as dissociation constant by SPR methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50625919(CHEMBL5431301)
Affinity DataKd:  722nMAssay Description:Binding affinity to his tagged BRDT bromodomain (unknown origin) assessed as dissociation constant by SPR methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetBromodomain testis-specific protein(Human)
Baylor College of Medicine

Curated by ChEMBL
LigandPNGBDBM50625920(CHEMBL5414263)
Affinity DataKd:  3.92E+3nMAssay Description:Binding affinity to his tagged BRDT bromodomain (unknown origin) assessed as dissociation constant by SPR methodMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed