Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50022380
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sapienza University of Rome
Curated by ChEMBL
Sapienza University of Rome
Curated by ChEMBL
Affinity DataKd: 690nMAssay Description:Binding affinity to human SIRT3 assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sapienza University of Rome
Curated by ChEMBL
Sapienza University of Rome
Curated by ChEMBL
Affinity DataKd: 3.90E+3nMAssay Description:Binding affinity to human SIRT3 (102 to 399 residues) expressed in Escherichia coli BL21 (DE3) cells assessed as dissociation constantMore data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Human)
Sapienza University of Rome
Curated by ChEMBL
Sapienza University of Rome
Curated by ChEMBL
Affinity DataIC50: 7.58E+4nMAssay Description:Activation of human SIRT3 (unknown origin) deacetylation activity using fluorogenic substrate measured upto 120 mins by microplate reader analysisMore data for this Ligand-Target Pair

