Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50020082
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50626021(CHEMBL5431205)
Affinity DataIC50: 55nMAssay Description:Inhibition of human TAK1 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50626020(CHEMBL5417075)
Affinity DataIC50: 63nMAssay Description:Inhibition of human TAK1 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50626019(CHEMBL5408799)
Affinity DataIC50: 83nMAssay Description:Inhibition of human TAK1 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50626026(CHEMBL5412383)
Affinity DataIC50: 116nMAssay Description:Inhibition of human TAK1 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50626024(CHEMBL5424789)
Affinity DataIC50: 131nMAssay Description:Inhibition of human TAK1 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50626027(CHEMBL5398734)
Affinity DataIC50: 172nMAssay Description:Inhibition of human TAK1 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50626029(CHEMBL5414193)
Affinity DataIC50: 187nMAssay Description:Inhibition of human TAK1 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50626028(CHEMBL5405261)
Affinity DataIC50: 192nMAssay Description:Inhibition of human TAK1 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50626025(CHEMBL5424167)
Affinity DataIC50: 199nMAssay Description:Inhibition of human TAK1 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50626022(CHEMBL5400329)
Affinity DataIC50: 205nMAssay Description:Inhibition of human TAK1 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50626023(CHEMBL5424796)
Affinity DataIC50: 208nMAssay Description:Inhibition of human TAK1 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed