Compile Data Set for Download or QSAR
Report error Found 130 Enz. Inhib. hit(s) with all data for entry = 50021446
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM220447(US9296741, 36 | US10633379, Compound X)
Affinity DataKd:  3nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640750(CHEMBL5575133)
Affinity DataIC50: 3.5nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640749(CHEMBL5572793 | US20250304550, Compound 4)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640762(CHEMBL5564568)
Affinity DataIC50: 7nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640752(CHEMBL5569832)
Affinity DataKd:  8.10nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640768(CHEMBL5589873)
Affinity DataKd:  8.90nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain testis-specific protein(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640768(CHEMBL5589873)
Affinity DataKd:  10nMAssay Description:Binding affinity to BRDT BD1 (unknown origin) assessed as dissociation constant by BROMOscan analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640769(CHEMBL5571807)
Affinity DataKd:  10nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640768(CHEMBL5589873)
Affinity DataKd:  10nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) assessed as dissociation constant by BROMOscan analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640765(CHEMBL5564917)
Affinity DataIC50: 11nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640761(CHEMBL5575268)
Affinity DataIC50: 11nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640764(CHEMBL5593751)
Affinity DataIC50: 12nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640769(CHEMBL5571807)
Affinity DataIC50: 12nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640768(CHEMBL5589873)
Affinity DataIC50: 12nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM220447(US9296741, 36 | US10633379, Compound X)
Affinity DataKd:  14nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 3(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640768(CHEMBL5589873)
Affinity DataKd:  14nMAssay Description:Binding affinity to BRD3 BD1 (unknown origin) assessed as dissociation constant by BROMOscan analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640752(CHEMBL5569832)
Affinity DataIC50: 15nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640750(CHEMBL5575133)
Affinity DataIC50: 16nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD2 incubated for 15 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640763(CHEMBL5570677)
Affinity DataIC50: 16nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640773(CHEMBL5568860)
Affinity DataIC50: 16nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640752(CHEMBL5569832)
Affinity DataIC50: 16nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD2 incubated for 15 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640760(CHEMBL5572940)
Affinity DataIC50: 18nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640762(CHEMBL5564568)
Affinity DataKd:  19nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640750(CHEMBL5575133)
Affinity DataKd:  20nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640756(CHEMBL5564525)
Affinity DataIC50: 22nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640764(CHEMBL5593751)
Affinity DataKd:  28nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 2(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640768(CHEMBL5589873)
Affinity DataKd:  28nMAssay Description:Binding affinity to BRD2 BD1 (unknown origin) assessed as dissociation constant by BROMOscan analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640771(CHEMBL5570515)
Affinity DataIC50: 28nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataIC50: 30nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640763(CHEMBL5570677)
Affinity DataKd:  31nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640757(CHEMBL5574846)
Affinity DataKd:  39nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640751(CHEMBL5573825)
Affinity DataKd:  41nMAssay Description:Binding affinity to his-tagged human BRD4 BD2 assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50544597(GSK778)
Affinity DataIC50: 41nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640756(CHEMBL5564525)
Affinity DataKd:  41nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640750(CHEMBL5575133)
Affinity DataKd:  41nMAssay Description:Binding affinity to his-tagged human BRD4 BD2 assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640760(CHEMBL5572940)
Affinity DataKd:  46nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  49nMAssay Description:Binding affinity to BRD4 BD1 (unknown origin) by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50544300(GSK046)
Affinity DataIC50: 49nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640757(CHEMBL5574846)
Affinity DataIC50: 56nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640759(CHEMBL5575904)
Affinity DataKd:  60nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640765(CHEMBL5564917)
Affinity DataKd:  61nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640772(CHEMBL5570353)
Affinity DataIC50: 69nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640758(CHEMBL5570823)
Affinity DataIC50: 74nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50543359(GSK620)
Affinity DataIC50: 81nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640774(CHEMBL5573799)
Affinity DataKd:  82nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640774(CHEMBL5573799)
Affinity DataIC50: 85nMAssay Description:Inhibition of N-terminal his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells incubated for 15 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640762(CHEMBL5564568)
Affinity DataKd:  90nMAssay Description:Binding affinity to his-tagged human BRD4 BD2 assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50640771(CHEMBL5570515)
Affinity DataKd:  94nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  95nMAssay Description:Binding affinity to his6-tagged human BRD4 BD1 (44 to 168 residues) expressed in Escherichia coli Rossetta BL21 (DE3) cells assessed as dissociation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50365262(CHEMBL1957266 | (S)-JQ1 (1) | US9320741, (S)-JQ1 |...)
Affinity DataKd:  96nMAssay Description:Binding affinity to BRD4 BD2 (unknown origin) by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
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