Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50021655
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
Shandong First Medical University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 11nMAssay Description:Inhibition of MNK2 (unknown origin) incubated for 60 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Human)
Shandong First Medical University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 49nMAssay Description:Inhibition of MNK1 (unknown origin) incubated for 60 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Human)
Shandong First Medical University

Curated by ChEMBL
LigandPNGBDBM50643127(CHEMBL5590391)
Affinity DataIC50: 121nMAssay Description:Inhibition of MNK1 (unknown origin) incubated for 60 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
Shandong First Medical University

Curated by ChEMBL
LigandPNGBDBM50643127(CHEMBL5590391)
Affinity DataIC50: 135nMAssay Description:Inhibition of MNK2 (unknown origin) incubated for 60 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
Shandong First Medical University

Curated by ChEMBL
LigandPNGBDBM50643126(CHEMBL5574018)
Affinity DataIC50: 199nMAssay Description:Inhibition of MNK2 (unknown origin) incubated for 60 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Human)
Shandong First Medical University

Curated by ChEMBL
LigandPNGBDBM50643126(CHEMBL5574018)
Affinity DataIC50: 401nMAssay Description:Inhibition of MNK1 (unknown origin) incubated for 60 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
Shandong First Medical University

Curated by ChEMBL
LigandPNGBDBM50643125(CHEMBL5566363)
Affinity DataIC50: 575nMAssay Description:Inhibition of MNK2 (unknown origin) incubated for 60 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
Shandong First Medical University

Curated by ChEMBL
LigandPNGBDBM50643124(CHEMBL5568981)
Affinity DataIC50: 587nMAssay Description:Inhibition of MNK2 (unknown origin) incubated for 60 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Human)
Shandong First Medical University

Curated by ChEMBL
LigandPNGBDBM50643125(CHEMBL5566363)
Affinity DataIC50: 596nMAssay Description:Inhibition of MNK1 (unknown origin) incubated for 60 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Human)
Shandong First Medical University

Curated by ChEMBL
LigandPNGBDBM50643124(CHEMBL5568981)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of MNK1 (unknown origin) incubated for 60 mins in presence of ATP by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed