Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50021031
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Cytokinetics, Inc.

Curated by ChEMBL
LigandPNGBDBM50636134(CHEMBL5558765)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of PDE3A (unknown origin) using cAMP as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by HTS as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Cytokinetics, Inc.

Curated by ChEMBL
LigandPNGBDBM50636136(CHEMBL5568428)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of PDE3A (unknown origin) using cAMP as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by HTS as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Cytokinetics, Inc.

Curated by ChEMBL
LigandPNGBDBM50636135(CHEMBL5566201)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of PDE3A (unknown origin) using cAMP as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by HTS as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Cytokinetics, Inc.

Curated by ChEMBL
LigandPNGBDBM50636138(CHEMBL5567433)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of PDE3A (unknown origin) using cAMP as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by HTS as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Cytokinetics, Inc.

Curated by ChEMBL
LigandPNGBDBM50636137(CHEMBL5558245)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of PDE3A (unknown origin) using cAMP as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by HTS as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Cytokinetics, Inc.

Curated by ChEMBL
LigandPNGBDBM50636140(CHEMBL5537058)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of PDE3A (unknown origin) using cAMP as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by HTS as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Cytokinetics, Inc.

Curated by ChEMBL
LigandPNGBDBM50636139(CHEMBL5542554)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of PDE3A (unknown origin) using cAMP as substrate preincubated for 20 mins followed by substrate addition measured after 30 mins by HTS as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetCytochrome P450 2A2(Rat)
Cytokinetics, Inc.

Curated by ChEMBL
LigandPNGBDBM50469700(CHEBI:50567 | (-)-OR-1259 | Levosimendan | OR-1259...)
Affinity DataKd:  1.00E+5nMAssay Description:Binding affinity to recombinant human Cardiac troponin C (1 to 89 residues) expressed in Escherichia coli assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed