Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50021487
TargetSolute carrier family 22 member 12(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50641286(CHEMBL5590320)
Affinity DataIC50: 2.01E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293T cells using 14C- uric acid assessed as uric acid absorption by measuring intracellular liquid radiatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50641281(CHEMBL5542414)
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293T cells using 14C- uric acid assessed as uric acid absorption by measuring intracellular liquid radiatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50641285(CHEMBL5579679)
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293T cells using 14C- uric acid assessed as uric acid absorption by measuring intracellular liquid radiatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50641288(CHEMBL5570059)
Affinity DataIC50: 3.75E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293T cells using 14C- uric acid assessed as uric acid absorption by measuring intracellular liquid radiatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50641287(CHEMBL5565332)
Affinity DataIC50: 3.96E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293T cells using 14C- uric acid assessed as uric acid absorption by measuring intracellular liquid radiatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50641283(CHEMBL5555561)
Affinity DataIC50: 4.35E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293T cells using 14C- uric acid assessed as uric acid absorption by measuring intracellular liquid radiatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50641282(CHEMBL5573620)
Affinity DataIC50: 4.73E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293T cells using 14C- uric acid assessed as uric acid absorption by measuring intracellular liquid radiatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50641284(CHEMBL5571882)
Affinity DataIC50: 4.86E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293T cells using 14C- uric acid assessed as uric acid absorption by measuring intracellular liquid radiatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSolute carrier family 22 member 12(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM37953(US10093631, Compound Lesinurad | US10336710, Lesin...)
Affinity DataIC50: 5.54E+3nMAssay Description:Inhibition of human URAT1 expressed in HEK293T cells using 14C- uric acid assessed as uric acid absorption by measuring intracellular liquid radiatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 9(Mus musculus)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50641286(CHEMBL5590320)
Affinity DataIC50: 1.82E+4nMAssay Description:Inhibition of mouse EGFP-tagged GLUT9 expressed in HEK293T cells assessed as inhibition rate by measuring relative current by patch clamp electrophys...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed