Compile Data Set for Download or QSAR
Report error Found 81 Enz. Inhib. hit(s) with all data for entry = 50021038
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM177922(US9675614, 166 | US10307413, Compound 337 | US1039...)
Affinity DataIC50: 47nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 62nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636262(CHEMBL5555046)
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636262(CHEMBL5555046)
Affinity DataIC50: 1.93E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636251(CHEMBL5532212)
Affinity DataIC50: 2.13E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636260(CHEMBL5560327)
Affinity DataIC50: 2.32E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636248(CHEMBL5557733)
Affinity DataIC50: 2.54E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636247(CHEMBL5542156)
Affinity DataIC50: 3.24E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636254(CHEMBL5562728)
Affinity DataIC50: 3.68E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636255(CHEMBL5555183)
Affinity DataIC50: 4.13E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636244(CHEMBL5556316)
Affinity DataIC50: 4.27E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636248(CHEMBL5557733)
Affinity DataIC50: 4.28E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636227(CHEMBL5558214)
Affinity DataIC50: 4.63E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636259(CHEMBL5559904)
Affinity DataIC50: 4.69E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636244(CHEMBL5556316)
Affinity DataIC50: 4.87E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636255(CHEMBL5555183)
Affinity DataIC50: 5.14E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636243(CHEMBL5562868)
Affinity DataIC50: 5.15E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636251(CHEMBL5532212)
Affinity DataIC50: 5.20E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636257(CHEMBL5560045)
Affinity DataIC50: 5.56E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636249(CHEMBL5555783)
Affinity DataIC50: 5.57E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636221(CHEMBL5566021)
Affinity DataIC50: 5.63E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636243(CHEMBL5562868)
Affinity DataIC50: 5.97E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636232(CHEMBL5560662)
Affinity DataIC50: 6.03E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636259(CHEMBL5559904)
Affinity DataIC50: 6.24E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636235(CHEMBL5555518)
Affinity DataIC50: 6.64E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636256(CHEMBL5568100)
Affinity DataIC50: 7.04E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636225(CHEMBL5563782)
Affinity DataIC50: 7.18E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636230(CHEMBL5562124)
Affinity DataIC50: 7.37E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636254(CHEMBL5562728)
Affinity DataIC50: 7.44E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636221(CHEMBL5566021)
Affinity DataIC50: 7.45E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636253(CHEMBL5561694)
Affinity DataIC50: 7.64E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636232(CHEMBL5560662)
Affinity DataIC50: 7.89E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636256(CHEMBL5568100)
Affinity DataIC50: 8.06E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636252(CHEMBL5567680)
Affinity DataIC50: 8.58E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-4(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636262(CHEMBL5555046)
Affinity DataIC50: 8.65E+4nMAssay Description:Inhibition of wild type GST-tagged HER4 catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636230(CHEMBL5562124)
Affinity DataIC50: 8.73E+4nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetHistone-arginine methyltransferase CARM1(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636262(CHEMBL5555046)
Affinity DataIC50: 8.76E+4nMAssay Description:Inhibition of PRMT4 (unknown origin) preincubated for 15 mins followed by substrate addition and measured after 60 mins by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636246(CHEMBL5523558)
Affinity DataIC50: 8.77E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetEpidermal growth factor receptor(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636225(CHEMBL5563782)
Affinity DataIC50: 9.52E+4nMAssay Description:Inhibition of wild type GST-tagged EGFR catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636262(CHEMBL5555046)
Affinity DataIC50: 9.82E+4nMAssay Description:Inhibition of wild type GST-tagged HER2 catalytic domain (unknown origin) expressed in insect cells using poly(Glu-Tyr) as substrate incubated for 6 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636242(CHEMBL5560064)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636241(CHEMBL5532149)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636240(CHEMBL5531979)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636239(CHEMBL5568227)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636245(CHEMBL5568296)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636246(CHEMBL5523558)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636252(CHEMBL5567680)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636250(CHEMBL5555395)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636226(CHEMBL5562615)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 5(Human)
Shandong University

Curated by ChEMBL
LigandPNGBDBM50636224(CHEMBL5512570)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT5 (unknown origin) by radiometric-based scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
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