Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50019644
TargetCREB-binding protein(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50100316(CHEMBL3321809)
Affinity DataIC50: 300nMAssay Description:Inhibition of CREBBP (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50598851(CHEMBL5199076 | US20240207300, Compound 292)
Affinity DataIC50: 300nMAssay Description:Inhibition of CREBBP (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetEphrin type-B receptor 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50154564(CHEMBL3774835 | US10688093, Compound DT2012-037541...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human EPHB4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetCasein kinase II subunit alpha(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50185757(CHEMBL3823403)
Affinity DataIC50: 500nMAssay Description:Inhibition of CK2alpha (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetEphrin type-B receptor 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50393033(CHEMBL2152699)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of human EPHB4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetBromodomain-containing protein 4(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50015249(CHEMBL1620811)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of BRD4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetTyrosine-protein kinase SYK(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50449315(CHEMBL3125863)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of SYK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetCREB-binding protein(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50172107(CHEMBL3810303)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of CREBBP (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMedPDB3D3D Structure (crystal)