Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50021745
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644403BDBM50644403(CHEMBL5564044)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644402BDBM50644402(CHEMBL5568986)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644399BDBM50644399(CHEMBL5573450)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50308135BDBM50308135(PKI-587 | 1-(4-{[4-(Dimethylamino)piperidin-1-yl]c...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644404BDBM50644404(CHEMBL5590872)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644398BDBM50644398(CHEMBL5566586)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644400BDBM50644400(CHEMBL5594441)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644392BDBM50644392(CHEMBL5568982)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644401BDBM50644401(CHEMBL5568655)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644415BDBM50644415(CHEMBL5575534)
Affinity DataIC50: 4nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644408BDBM50644408(CHEMBL5570798)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644410BDBM50644410(CHEMBL5570177)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644393BDBM50644393(CHEMBL5575213)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644409BDBM50644409(CHEMBL5567159)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644395BDBM50644395(CHEMBL5573179)
Affinity DataIC50: 5nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50308135BDBM50308135(PKI-587 | 1-(4-{[4-(Dimethylamino)piperidin-1-yl]c...)
Affinity DataIC50: 6nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644396BDBM50644396(CHEMBL5572519)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644394BDBM50644394(CHEMBL5570389)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644412BDBM50644412(CHEMBL5575407)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644398BDBM50644398(CHEMBL5566586)
Affinity DataIC50: 10nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644390BDBM50644390(CHEMBL5573982)
Affinity DataIC50: 11nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644396BDBM50644396(CHEMBL5572519)
Affinity DataIC50: 12nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644395BDBM50644395(CHEMBL5573179)
Affinity DataIC50: 15nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644414BDBM50644414(CHEMBL5590918)
Affinity DataIC50: 20nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644390BDBM50644390(CHEMBL5573982)
Affinity DataIC50: 22nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644395BDBM50644395(CHEMBL5573179)
Affinity DataIC50: 26nMAssay Description:Inhibition of PI3Kgamma (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50308135BDBM50308135(PKI-587 | 1-(4-{[4-(Dimethylamino)piperidin-1-yl]c...)
Affinity DataIC50: 28nMAssay Description:Inhibition of PI3Kbeta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644405BDBM50644405(CHEMBL5564938)
Affinity DataIC50: 29nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644389BDBM50644389(CHEMBL5567165)
Affinity DataIC50: 31nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644413BDBM50644413(CHEMBL5569846)
Affinity DataIC50: 32nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644397BDBM50644397(CHEMBL5566351)
Affinity DataIC50: 35nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644393BDBM50644393(CHEMBL5575213)
Affinity DataIC50: 38nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50308135BDBM50308135(PKI-587 | 1-(4-{[4-(Dimethylamino)piperidin-1-yl]c...)
Affinity DataIC50: 41nMAssay Description:Inhibition of PI3Kgamma (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644401BDBM50644401(CHEMBL5568655)
Affinity DataIC50: 44nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644394BDBM50644394(CHEMBL5570389)
Affinity DataIC50: 45nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644392BDBM50644392(CHEMBL5568982)
Affinity DataIC50: 45nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644387BDBM50644387(CHEMBL5574430)
Affinity DataIC50: 48nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644386BDBM50644386(CHEMBL5572006)
Affinity DataIC50: 53nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644400BDBM50644400(CHEMBL5594441)
Affinity DataIC50: 64nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644397BDBM50644397(CHEMBL5566351)
Affinity DataIC50: 75nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644401BDBM50644401(CHEMBL5568655)
Affinity DataIC50: 93nMAssay Description:Inhibition of PI3Kbeta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644395BDBM50644395(CHEMBL5573179)
Affinity DataIC50: 98nMAssay Description:Inhibition of PI3Kdelta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644389BDBM50644389(CHEMBL5567165)
Affinity DataIC50: 112nMAssay Description:Inhibition of PI3Kalpha (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644407BDBM50644407(CHEMBL5573360)
Affinity DataIC50: 116nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644392BDBM50644392(CHEMBL5568982)
Affinity DataIC50: 129nMAssay Description:Inhibition of PI3Kbeta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Guizhou Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50644411BDBM50644411(CHEMBL5575205)
Affinity DataIC50: 147nMAssay Description:Inhibition of mTOR (unknown origin) by Lance ultra assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50308135BDBM50308135(PKI-587 | 1-(4-{[4-(Dimethylamino)piperidin-1-yl]c...)
Affinity DataIC50: 156nMAssay Description:Inhibition of PI3Kdelta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644400BDBM50644400(CHEMBL5594441)
Affinity DataIC50: 157nMAssay Description:Inhibition of PI3Kbeta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644401BDBM50644401(CHEMBL5568655)
Affinity DataIC50: 161nMAssay Description:Inhibition of PI3Kdelta (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
LigandChemical structure of BindingDB Monomer ID 50644392BDBM50644392(CHEMBL5568982)
Affinity DataIC50: 162nMAssay Description:Inhibition of PI3Kgamma (unknown origin) by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
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