Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50021082
TargetC-C chemokine receptor type 6(Mus musculus)
Idorsia Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50636598(CHEMBL5561521)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at CCR6 in C57BL/6J mouse whole blood assessed as inhibition of CCL20-stimulated receptor internalization in lymphocytes incubate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetC-C chemokine receptor type 6(Human)
Idorsia Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50636599(CHEMBL5563681)
Affinity DataKi:  45nMAssay Description:Insurmountable antagonist activity at human CCR6 expressed in HEK293 cells co-transfected with firefly luciferase gene assessed as inhibition of CCL2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetATP-dependent translocase ABCB1(Human)
Idorsia Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50636599(CHEMBL5563681)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of human MDR1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSolute carrier organic anion transporter family member 1B3(Human)
Idorsia Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50636599(CHEMBL5563681)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of OATP1B3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetSolute carrier organic anion transporter family member 1B1(Human)
Idorsia Pharmaceuticals Ltd.

Curated by ChEMBL
LigandPNGBDBM50636599(CHEMBL5563681)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of OATP1B1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed