Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50021100
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50155926(CHEMBL3183703)
Affinity DataKd:  0.532nMAssay Description:Binding affinity to NLRP3 (unknown origin) expressed in HEK293T cells incubated for 30 mins by MST assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50155926(CHEMBL3183703)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of NLRP3 inflammasome activation in mouse BMDM preincubated with LPS for 3 hrs followed by compound addition for 30 mins and further stimu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50155926(CHEMBL3183703)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636762(CHEMBL5567870)
Affinity DataKd:  11nMAssay Description:Binding affinity to NLRP3 (unknown origin) expressed in HEK293T cells incubated for 30 mins by MST assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636753(Emlenoflast | Inzomelid | Izd-174 | Izd174 | MCC-7...)
Affinity DataIC50: 14nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636758(CHEMBL5561914)
Affinity DataIC50: 50nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636778(CHEMBL5562815)
Affinity DataIC50: 72nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636762(CHEMBL5567870)
Affinity DataIC50: 77nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636760(CHEMBL5564626)
Affinity DataIC50: 81nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636763(CHEMBL5568569)
Affinity DataIC50: 82nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636767(CHEMBL5567872)
Affinity DataIC50: 91nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636756(CHEMBL5560738)
Affinity DataIC50: 97nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636779(CHEMBL5565134)
Affinity DataIC50: 99nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636757(CHEMBL5542263)
Affinity DataIC50: 99nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636780(CHEMBL5561461)
Affinity DataIC50: 100nMAssay Description:Inhibition of NLRP3 inflammasome activation in mouse J774.A1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636755(CHEMBL5560910)
Affinity DataIC50: 100nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636769(CHEMBL5555459)
Affinity DataIC50: 102nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636770(CHEMBL5556291)
Affinity DataIC50: 103nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636768(CHEMBL5542299)
Affinity DataIC50: 137nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636773(CHEMBL5566190)
Affinity DataIC50: 137nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636777(CHEMBL5542998)
Affinity DataIC50: 147nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636776(CHEMBL5555806)
Affinity DataIC50: 161nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636771(CHEMBL5555591)
Affinity DataIC50: 178nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636774(CHEMBL5557207)
Affinity DataIC50: 195nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636764(CHEMBL5561902)
Affinity DataIC50: 216nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636754(CHEMBL5560131)
Affinity DataIC50: 232nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636772(CHEMBL5556036)
Affinity DataIC50: 242nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636765(CHEMBL5560261)
Affinity DataIC50: 283nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636766(CHEMBL5542234)
Affinity DataIC50: 286nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636775(CHEMBL5560697)
Affinity DataIC50: 292nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636761(CHEMBL5542903)
Affinity DataIC50: 406nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50605174(CHEMBL1164920)
Affinity DataIC50: 780nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50636759(CHEMBL5532284)
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in LPS/ATP-induced C57BL/6 mouse BMDMs assessed as reduction in IL-1beta secretion preincubated with LPS ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50505851(CHEMBL4583133)
Affinity DataIC50: 8.45E+3nMAssay Description:Inhibition of NLRP3 inflammasome activation in mouse J774.A1 cells preincubated with LPS for 4.5 hrs followed by compound addition for 30 mins and fu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50012957(1-((p-(2-(5-chloro-o-anisamido)ethyl)phenyl)sulfon...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 inflammasome activation in mouse BMDMsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50372524(BAY-11-7082 | CHEMBL403183)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of mouse NLRP3 inflammasome expressed in NG5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed