Compile Data Set for Download or QSAR
Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 50020962
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635542(CHEMBL5557729)
Affinity DataEC50:  46nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635554(CHEMBL5556102)
Affinity DataEC50:  54nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635555(CHEMBL5555231)
Affinity DataEC50:  58nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635562(CHEMBL5523402)
Affinity DataEC50:  90nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635561(CHEMBL5532000)
Affinity DataEC50:  121nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635553(CHEMBL5558124)
Affinity DataEC50:  124nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635565(CHEMBL5556346)
Affinity DataEC50:  127nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635535(CHEMBL5557995)
Affinity DataEC50:  128nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635545(CHEMBL5542965)
Affinity DataEC50:  150nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)TBA
LigandPNGBDBM50635545(CHEMBL5542965)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant by radioligand competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635537(CHEMBL5555055)
Affinity DataEC50:  156nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635536(CHEMBL5556677)
Affinity DataEC50:  157nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635563(CHEMBL5557839)
Affinity DataEC50:  161nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635544(CHEMBL5557393)
Affinity DataEC50:  171nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635540(CHEMBL5517636)
Affinity DataEC50:  180nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635534(CHEMBL5505829)
Affinity DataEC50:  194nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635527(CHEMBL5558263)
Affinity DataEC50:  207nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635543(CHEMBL5549936)
Affinity DataEC50:  216nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635539(CHEMBL5512594)
Affinity DataEC50:  220nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635567(CHEMBL5556049)
Affinity DataEC50:  230nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635557(CHEMBL5559512)
Affinity DataEC50:  241nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635560(CHEMBL5532256)
Affinity DataEC50:  244nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635541(CHEMBL5523442)
Affinity DataEC50:  245nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635564(CHEMBL5555914)
Affinity DataEC50:  251nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635556(CHEMBL5556617)
Affinity DataEC50:  280nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635558(CHEMBL5557780)
Affinity DataEC50:  281nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635566(CHEMBL5559109)
Affinity DataEC50:  288nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635570(CHEMBL5556551)
Affinity DataEC50:  290nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635571(CHEMBL5557906)
Affinity DataEC50:  297nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635526(CHEMBL5517653)
Affinity DataEC50:  299nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635538(CHEMBL5542310)
Affinity DataEC50:  301nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635531(CHEMBL5523497)
Affinity DataEC50:  318nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635568(CHEMBL5558536)
Affinity DataEC50:  334nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)TBA
LigandPNGBDBM50635540(CHEMBL5517636)
Affinity DataKi:  344nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant by radioligand competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635532(CHEMBL5505756)
Affinity DataEC50:  371nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635528(CHEMBL5505898)
Affinity DataEC50:  379nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635525(CHEMBL5517700)
Affinity DataEC50:  379nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635577(CHEMBL5558192)
Affinity DataEC50:  393nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635576(CHEMBL5556254)
Affinity DataEC50:  398nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635569(CHEMBL5558126)
Affinity DataEC50:  444nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635530(CHEMBL5558903)
Affinity DataEC50:  447nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)TBA
LigandPNGBDBM50635554(CHEMBL5556102)
Affinity DataKi:  481nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant by radioligand competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635546(CHEMBL5557185)
Affinity DataEC50:  488nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635559(CHEMBL5527882)
Affinity DataEC50:  559nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50561705(CHEMBL4758188)
Affinity DataEC50:  582nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635575(CHEMBL5523663)
Affinity DataEC50:  711nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)TBA
LigandPNGBDBM50635542(CHEMBL5557729)
Affinity DataKi:  827nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant by radioligand competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)TBA
LigandPNGBDBM50635539(CHEMBL5512594)
Affinity DataKi:  896nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in CHO cells assessed as inhibition constant by radioligand competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetN-arachidonyl glycine receptor(Mus musculus)TBA
LigandPNGBDBM50635572(CHEMBL5556616)
Affinity DataEC50:  981nMAssay Description:Agonist activity at mouse GPR18 expressed in CHO cells assessed as activation by measuring beta-arrestin2 recruitment incubated for 90 mins by lumine...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)TBA
LigandPNGBDBM50635554(CHEMBL5556102)
Affinity DataKi:  1.18E+3nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in CHO cells assessed as inhibition constant by radioligand competition binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
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