Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50021395
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640163(CHEMBL5568491)
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640152(CHEMBL5561987)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640153(CHEMBL5532138)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640160(CHEMBL5561563)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640164(CHEMBL5563634)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640162(CHEMBL5560073)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640161(CHEMBL5561245)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640157(CHEMBL5562881)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50601904(CHEMBL5184663)
Affinity DataIC50: 5.70nMAssay Description:Inhibition of Plasmodium falciparum SUB1More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640167(CHEMBL5567696)
Affinity DataIC50: 6nMAssay Description:Inhibition of human 20s proteasome beta5 subunit mediated chymotrypsin-like activity using LLVY-R110 as substrate measured every three mins for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640155(CHEMBL5564605)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640159(CHEMBL5561949)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640169(CHEMBL5565717)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640168(CHEMBL5556185)
Affinity DataIC50: 7nMAssay Description:Inhibition of human 20s proteasome beta5 subunit mediated chymotrypsin-like activity using LLVY-R110 as substrate measured every three mins for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640154(CHEMBL5563835)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640158(CHEMBL5559405)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50601901(CHEMBL5180525)
Affinity DataIC50: 9.30nMAssay Description:Inhibition of Plasmodium falciparum SUB1More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640168(CHEMBL5556185)
Affinity DataIC50: 9.30nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640167(CHEMBL5567696)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640171(CHEMBL5562284)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640172(CHEMBL5567647)
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640173(CHEMBL5564621)
Affinity DataIC50: 19nMAssay Description:Inhibition of Plasmodium falciparum SUB1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640165(CHEMBL5561366)
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50601904(CHEMBL5184663)
Affinity DataIC50: 33nMAssay Description:Inhibition of human 20s proteasome beta5 subunit mediated chymotrypsin-like activity using LLVY-R110 as substrate measured every three mins for 1 hr ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50601901(CHEMBL5180525)
Affinity DataIC50: 35nMAssay Description:Inhibition of human 20s proteasome beta5 subunit mediated chymotrypsin-like activity using LLVY-R110 as substrate measured every three mins for 1 hr ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640170(CHEMBL5561760)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640156(CHEMBL5555306)
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetSubtilisin-like protease 1(malaria parasite P. falciparum)TBA
LigandPNGBDBM50640166(CHEMBL5565877)
Affinity DataIC50: 71nMAssay Description:Inhibition of recombinant Plasmodium falciparum SUB1 using Ac-CKITAQDDEESC-OH as fluorogenic substrate pre-incubated for 5 mins followed by substrate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640171(CHEMBL5562284)
Affinity DataIC50: 160nMAssay Description:Inhibition of human 20s proteasome beta5 subunit mediated chymotrypsin-like activity using LLVY-R110 as substrate measured every three mins for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640170(CHEMBL5561760)
Affinity DataIC50: 410nMAssay Description:Inhibition of human 20s proteasome beta5 subunit mediated chymotrypsin-like activity using LLVY-R110 as substrate measured every three mins for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640172(CHEMBL5567647)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human 20s proteasome beta5 subunit mediated chymotrypsin-like activity using LLVY-R110 as substrate measured every three mins for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640173(CHEMBL5564621)
Affinity DataIC50: 3.56E+4nMAssay Description:Inhibition of human 20s proteasome beta5 subunit mediated chymotrypsin-like activity using LLVY-R110 as substrate measured every three mins for 1 hr ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed