Compile Data Set for Download or QSAR
Report error Found 69 Enz. Inhib. hit(s) with all data for entry = 50021397
LigandPNGBDBM720656((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720664((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640191(CHEMBL5550050)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720659((R)-4-(2-(1H-indol-4-yl)-7-(methylsulfonyl)-7H-pyr...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720656((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human ATRMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640175(CHEMBL5567922)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640184(CHEMBL5566930)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640182(CHEMBL5563958)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720687((R)-4-(2-(6-chloro-1H-indol-4-yl)-7-(methylsulfony...)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50427326(CHEMBL2325697)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720688((R)-4-(2-(6-methoxy-1H-indol-4-yl)-7-(methylsulfon...)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640185(CHEMBL5565708)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640181(CHEMBL5532143)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640176(CHEMBL5561105)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640180(CHEMBL5542235)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640183(CHEMBL5560533)
Affinity DataIC50: 8nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640192(CHEMBL5558671)
Affinity DataIC50: 9.20nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720686((R)-4-(4-(3-methylmorpholinyl)-7-(methylsulfonyl)-...)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640177(CHEMBL5561890)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720664((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 22nMAssay Description:Inhibition of human mTORMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640194(CHEMBL5564228)
Affinity DataIC50: 28nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640178(CHEMBL5566032)
Affinity DataIC50: 32nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640200(CHEMBL5561297)
Affinity DataIC50: 40nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640179(CHEMBL5568241)
Affinity DataIC50: 44nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720656((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 46nMAssay Description:Inhibition of human mTORMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640198(CHEMBL5562666)
Affinity DataIC50: 47nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640195(CHEMBL5568258)
Affinity DataIC50: 53nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640190(CHEMBL5560978)
Affinity DataIC50: 85nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720656((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 119nMAssay Description:Inhibition of human DNA-PKMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640186(CHEMBL5561408)
Affinity DataIC50: 205nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640196(CHEMBL5561516)
Affinity DataIC50: 245nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640187(CHEMBL5562160)
Affinity DataIC50: 270nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640197(CHEMBL5556934)
Affinity DataIC50: 625nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640201(CHEMBL5555066)
Affinity DataIC50: 630nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640193(CHEMBL5555314)
Affinity DataIC50: 684nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640174(CHEMBL5561060)
Affinity DataIC50: 746nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720656((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of human PI3KalphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720656((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 2.59E+3nMAssay Description:Inhibition of human LCKMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720656((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 3.21E+3nMAssay Description:Inhibition of human ATMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640188(CHEMBL5564689)
Affinity DataIC50: 3.67E+3nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM50640199(CHEMBL5558523)
Affinity DataIC50: 3.69E+3nMAssay Description:Inhibition of ATR/ATRIP (unknown origin) using 5-FAM-AK-17 as substrate preincubated with compound for 10 mins followed by ATP addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720664((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 4.95E+3nMAssay Description:Inhibition of human LCKMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720656((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 7.31E+3nMAssay Description:Inhibition of human ARK5More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720664((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human JAK1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720656((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human JAK1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetAurora kinase B(Human)TBA
LigandPNGBDBM720664((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human Aurora BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
TargetAurora kinase B(Human)TBA
LigandPNGBDBM720656((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human Aurora BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720664((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human AMPK alpha2/beta1/gamma1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720656((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human AMPK alpha2/beta1/gamma1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
LigandPNGBDBM720664((R)-3-methyl-4-(7-(methylsulfonyl)-2-(1H-pyrrolo[2...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CDK2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
PubMed
Displayed 1 to 50 (of 69 total ) | Next | Last >>
Jump to: