Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50022223
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649615(CHEMBL5618909)
Affinity DataKd:  60nMAssay Description:Binding affinity to human TLX LBD assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649609(CHEMBL5618548)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649612(CHEMBL5618740)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649595(CHEMBL5619615)
Affinity DataKd:  110nMAssay Description:Binding affinity to human TLX LBD assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649589(CHEMBL5619500)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649615(CHEMBL5618909)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649612(CHEMBL5618740)
Affinity DataKd:  160nMAssay Description:Binding affinity to human TLX LBD assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649604(CHEMBL5619514)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649597(CHEMBL5618246)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649595(CHEMBL5619615)
Affinity DataEC50:  260nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649604(CHEMBL5619514)
Affinity DataKd:  360nMAssay Description:Binding affinity to human TLX LBD assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649614(CHEMBL5619484)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649592(CHEMBL5618230)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649607(CHEMBL5618588)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649602(CHEMBL5619493)
Affinity DataEC50:  600nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649593(CHEMBL5618438)
Affinity DataEC50:  700nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649596(CHEMBL5620162)
Affinity DataEC50:  700nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649608(CHEMBL5618094)
Affinity DataEC50:  900nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649611(CHEMBL5618699)
Affinity DataEC50:  900nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649606(CHEMBL5618147)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649613(CHEMBL5619983)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649610(CHEMBL5620053)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649598(CHEMBL5618709)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-alpha(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649615(CHEMBL5618909)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of ROR-alpha (unknown origin) expressed in HEK293T cells co-transfected with RL/Gal4-VP16 incubated for 16 hrs by Dual-Glo Luciferase assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649594(CHEMBL5619707)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649605(CHEMBL5619135)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649603(CHEMBL5618526)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649590(CHEMBL5620146)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649599(CHEMBL5620263)
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649601(CHEMBL5618097)
Affinity DataEC50:  8.00E+3nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-alpha(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649612(CHEMBL5618740)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of ROR-alpha (unknown origin) expressed in HEK293T cells co-transfected with RL/Gal4-VP16 incubated for 16 hrs by Dual-Glo Luciferase assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649591(CHEMBL5619131)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor subfamily 2 group E member 1(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649600(CHEMBL5619639)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLX LBD expressed in HEK293T cells co-transfected with RL/Gal4-VP16 assessed as repression of VP16-induced reporter activit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear receptor ROR-alpha(Human)
Ludwig-Maximilians-Universitat (LMU) Munchen

Curated by ChEMBL
LigandPNGBDBM50649604(CHEMBL5619514)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ROR-alpha (unknown origin) expressed in HEK293T cells co-transfected with RL/Gal4-VP16 incubated for 16 hrs by Dual-Glo Luciferase assa...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed