Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50022004
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50155926BDBM50155926(CHEMBL3183703)
Affinity DataIC50: 12nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetNACHT, LRR and PYD domains-containing protein 3(Mouse)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647121BDBM50647121(CHEMBL5591066)
Affinity DataIC50: 210nMAssay Description:Inhibition of NLRP3 inflammasome activation in M-CSF induced C57BL/6 mouse BMDM cells assessed as inhibition of LPS/nigericin induced IL-1beta produc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647121BDBM50647121(CHEMBL5591066)
Affinity DataIC50: 260nMAssay Description:Inhibition of NLRP3 inflammasome activation in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta producti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647121BDBM50647121(CHEMBL5591066)
Affinity DataIC50: 260nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647123BDBM50647123(CHEMBL5591726)
Affinity DataIC50: 430nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647120BDBM50647120(CHEMBL5590770)
Affinity DataIC50: 680nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647119BDBM50647119(CHEMBL5590073)
Affinity DataIC50: 710nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647124BDBM50647124(CHEMBL5595030)
Affinity DataIC50: 810nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647117BDBM50647117(CHEMBL5590187)
Affinity DataIC50: 960nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647118BDBM50647118(CHEMBL5592068)
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647121BDBM50647121(CHEMBL5591066)
Affinity DataKd:  1.05E+3nMAssay Description:Binding affinity to human NLRP3 assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647088BDBM50647088(CHEMBL5596006)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647125BDBM50647125(CHEMBL5592969)
Affinity DataIC50: 1.88E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647074BDBM50647074(CHEMBL5593521)
Affinity DataIC50: 4.07E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647086BDBM50647086(CHEMBL5595876)
Affinity DataIC50: 4.31E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647122BDBM50647122(CHEMBL5595046)
Affinity DataIC50: 4.34E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647084BDBM50647084(CHEMBL5595175)
Affinity DataIC50: 4.42E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647116BDBM50647116(CHEMBL5592483)
Affinity DataIC50: 5.03E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647098BDBM50647098(CHEMBL5591774)
Affinity DataIC50: 5.19E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647077BDBM50647077(CHEMBL5592212)
Affinity DataIC50: 6.93E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647078BDBM50647078(CHEMBL5595491)
Affinity DataIC50: 7.31E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647087BDBM50647087(CHEMBL5593090)
Affinity DataIC50: 7.67E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647093BDBM50647093(CHEMBL5594085)
Affinity DataIC50: 7.88E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647082BDBM50647082(CHEMBL5593101)
Affinity DataIC50: 9.74E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647091BDBM50647091(CHEMBL5593950)
Affinity DataIC50: 9.89E+3nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647097BDBM50647097(CHEMBL5591887)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647096BDBM50647096(CHEMBL5594303)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647095BDBM50647095(CHEMBL5593730)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647102BDBM50647102(CHEMBL5592552)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647101BDBM50647101(CHEMBL5591402)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647100BDBM50647100(CHEMBL5592332)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647099BDBM50647099(CHEMBL5593527)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647106BDBM50647106(CHEMBL5590752)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647105BDBM50647105(CHEMBL5593105)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647104BDBM50647104(CHEMBL5592831)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647103BDBM50647103(CHEMBL5590482)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647110BDBM50647110(CHEMBL5594976)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647109BDBM50647109(CHEMBL5593889)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647108BDBM50647108(CHEMBL5589633)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647107BDBM50647107(CHEMBL5592142)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647081BDBM50647081(CHEMBL5590194)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647080BDBM50647080(CHEMBL5595666)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647079BDBM50647079(CHEMBL5593637)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647085BDBM50647085(CHEMBL5592767)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647083BDBM50647083(CHEMBL5594368)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647090BDBM50647090(CHEMBL5592777)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647089BDBM50647089(CHEMBL5594957)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647094BDBM50647094(CHEMBL5589977)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647092BDBM50647092(CHEMBL5583735)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetNACHT, LRR and PYD domains-containing protein 3(Human)
Fudan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50647076BDBM50647076(CHEMBL5595419)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of NLRP3 in PMA-differentiated human THP-1 cells assessed as inhibition of LPS/nigericin induced IL-1beta production by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
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