Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50023692
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666820BDBM50666820(CHEMBL6173629)
Affinity DataEC50:  120nMAssay Description:Activation of hyperactive human BKca channel G803D/N806K mutant transfected in human AD-293 cells incubated for 15 mins by Flexstation3 multimode mic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50426567BDBM50426567(BMS-204352 | MaxiPost | FLINDOKALNER)
Affinity DataEC50:  350nMAssay Description:Activation of human BKca channel expressed in HEK293 cells by patch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666827BDBM50666827(CHEMBL4303589)
Affinity DataEC50:  400nMAssay Description:Activation of human KCa1.1 by patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666823BDBM50666823(CHEMBL6166658)
Affinity DataEC50:  420nMAssay Description:Activation of hyperactive human BKca channel G803D/N806K mutant transfected in human AD-293 cells incubated for 15 mins by Flexstation3 multimode mic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666819BDBM50666819(CHEMBL6176092)
Affinity DataEC50:  680nMAssay Description:Activation of hyperactive human BKca channel G803D/N806K mutant transfected in human AD-293 cells incubated for 15 mins by Flexstation3 multimode mic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666821BDBM50666821(CHEMBL6166315)
Affinity DataEC50:  1.21E+3nMAssay Description:Activation of hyperactive human BKca channel G803D/N806K mutant transfected in human AD-293 cells incubated for 15 mins by Flexstation3 multimode mic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666822BDBM50666822(CHEMBL6169698)
Affinity DataEC50:  1.37E+3nMAssay Description:Activation of hyperactive human BKca channel G803D/N806K mutant transfected in human AD-293 cells incubated for 15 mins by Flexstation3 multimode mic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666818BDBM50666818(CHEMBL6177233)
Affinity DataEC50:  1.58E+3nMAssay Description:Activation of hyperactive human BKca channel G803D/N806K mutant transfected in human AD-293 cells incubated for 15 mins by Flexstation3 multimode mic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666828BDBM50666828(CHEMBL5187254)
Affinity DataEC50:  2.70E+3nMAssay Description:Activation of BKca channel (unknown origin) by cell based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666828BDBM50666828(CHEMBL5187254)
Affinity DataEC50:  2.70E+3nMAssay Description:Activation of BKca channel (unknown origin) by cell-based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666825BDBM50666825(CHEMBL6177852)
Affinity DataEC50:  2.82E+3nMAssay Description:Activation of hyperactive human BKca channel G803D/N806K mutant transfected in human AD-293 cells incubated for 15 mins by Flexstation3 multimode mic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666829BDBM50666829(CHEMBL6145166)
Affinity DataEC50:  3.90E+3nMAssay Description:Activation of hyperactive human BKca channel G803D/N806K mutant transfected in human AD-293 cells incubated for 20 to 30 mins by Flexstation3 multimo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666826BDBM50666826(CHEMBL4859302)
Affinity DataEC50:  5.40E+3nMAssay Description:Activation of BKca channel (unknown origin) by cell-based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666826BDBM50666826(CHEMBL4859302)
Affinity DataEC50:  5.40E+3nMAssay Description:Activation of BKca channel (unknown origin) by cell based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666827BDBM50666827(CHEMBL4303589)
Affinity DataEC50:  7.00E+3nMAssay Description:Activation of BKca channel (unknown origin) by cell-based fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666827BDBM50666827(CHEMBL4303589)
Affinity DataEC50:  7.00E+3nMAssay Description:Activation of BKca channel (unknown origin) by cell based methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50666824BDBM50666824(CHEMBL6173767)
Affinity DataEC50:  9.22E+3nMAssay Description:Activation of hyperactive human BKca channel G803D/N806K mutant transfected in human AD-293 cells incubated for 15 mins by Flexstation3 multimode mic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50347497BDBM50347497(CHEMBL384903)
Affinity DataEC50:  1.00E+4nMAssay Description:Activation of BKca channel (unknown origin) by patch-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetCalcium-activated potassium channel subunit alpha-1(Human)
Gwangju Institute of Science and Technology

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50158460BDBM50158460(cid_2333 | Benzbromarone | 3,5-dibromo-4-hydroxyph...)
Affinity DataEC50:  1.11E+5nMAssay Description:Activation of human BK ca channel expressed in CHO cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed