Report error Found 110 Enz. Inhib. hit(s) with all data for entry = 50023773
Affinity DataEC50: 3.30E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 3.50E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 3.70E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 3.80E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 4.40E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 4.50E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 4.70E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 4.80E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 5.10E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 5.70E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 6.20E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 7.10E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 8.10E+3nMAssay Description:Agonist activity at mouse STING expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured after 24 hrs incubation b...More data for this Ligand-Target Pair
Affinity DataEC50: 8.20E+3nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 8.80E+3nMAssay Description:Agonist activity at STING R232 mutant (unknown origin) expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured af...More data for this Ligand-Target Pair
Affinity DataEC50: 9.00E+3nMAssay Description:Agonist activity at STING R232 mutant (unknown origin) expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured af...More data for this Ligand-Target Pair
Affinity DataEC50: 9.30E+3nMAssay Description:Agonist activity at mouse STING expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured after 24 hrs incubation b...More data for this Ligand-Target Pair
Affinity DataEC50: 1.13E+4nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 1.19E+4nMAssay Description:Agonist activity at mouse STING expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured after 24 hrs incubation b...More data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+4nMAssay Description:Agonist activity at STING R232 mutant (unknown origin) expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured af...More data for this Ligand-Target Pair
Affinity DataEC50: 1.25E+4nMAssay Description:Agonist activity at mouse STING expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured after 24 hrs incubation b...More data for this Ligand-Target Pair
Affinity DataEC50: 1.30E+4nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 1.32E+4nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 1.33E+4nMAssay Description:Agonist activity at STING R232 mutant (unknown origin) expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured af...More data for this Ligand-Target Pair
Affinity DataEC50: 1.45E+4nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 1.57E+4nMAssay Description:Agonist activity at mouse STING expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured after 24 hrs incubation b...More data for this Ligand-Target Pair
Affinity DataEC50: 1.72E+4nMAssay Description:Agonist activity at STING R232 mutant (unknown origin) expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured af...More data for this Ligand-Target Pair
Affinity DataEC50: 1.84E+4nMAssay Description:Agonist activity at STING R232 mutant (unknown origin) expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured af...More data for this Ligand-Target Pair
Affinity DataEC50: 1.96E+4nMAssay Description:Agonist activity at STING R232 mutant (unknown origin) expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured af...More data for this Ligand-Target Pair
Affinity DataEC50: 1.98E+4nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+4nMAssay Description:Agonist activity at mouse STING expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured after 24 hrs incubation b...More data for this Ligand-Target Pair
Affinity DataIC50: 2.21E+4nMAssay Description:Binding affinity to wild type His-tagged STING (unknown origin) measured after 3 hrs incubation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.25E+4nMAssay Description:Binding affinity to wild type His-tagged STING (unknown origin) measured after 3 hrs incubation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.36E+4nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataIC50: 2.41E+4nMAssay Description:Binding affinity to wild type His-tagged STING (unknown origin) measured after 3 hrs incubation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.46E+4nMAssay Description:Binding affinity to wild type His-tagged STING (unknown origin) measured after 3 hrs incubation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.51E+4nMAssay Description:Agonist activity at mouse STING expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured after 24 hrs incubation b...More data for this Ligand-Target Pair
Affinity DataEC50: 2.53E+4nMAssay Description:Agonist activity at mouse STING expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured after 24 hrs incubation b...More data for this Ligand-Target Pair
Affinity DataEC50: 2.61E+4nMAssay Description:Agonist activity at STING R232 mutant (unknown origin) expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured af...More data for this Ligand-Target Pair
Affinity DataEC50: 2.65E+4nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+4nMAssay Description:Agonist activity at mouse STING expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured after 24 hrs incubation b...More data for this Ligand-Target Pair
Affinity DataEC50: 2.79E+4nMAssay Description:Agonist activity at mouse STING expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured after 24 hrs incubation b...More data for this Ligand-Target Pair
Affinity DataIC50: 2.87E+4nMAssay Description:Binding affinity to wild type His-tagged STING (unknown origin) measured after 3 hrs incubation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.03E+4nMAssay Description:Agonist activity at human STING in human THP1-Blue ISG cells measured after 24 hrs incubation by QUANTI-Blue based microplate readerMore data for this Ligand-Target Pair
Affinity DataEC50: 3.03E+4nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataIC50: 3.06E+4nMAssay Description:Binding affinity to wild type His-tagged STING (unknown origin) measured after 3 hrs incubation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.12E+4nMAssay Description:Binding affinity to wild type His-tagged STING (unknown origin) measured after 3 hrs incubation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30E+4nMAssay Description:Agonist activity at human STING HAQ variant in human THP1-Blue ISG cells assessed as fold change in stimulation activity measured after 24 hrs incuba...More data for this Ligand-Target Pair
Affinity DataEC50: 3.31E+4nMAssay Description:Agonist activity at STING R232 mutant (unknown origin) expressed in human THP1-Dual cells assessed as fold change in stimulation activity measured af...More data for this Ligand-Target Pair
Affinity DataIC50: 3.33E+4nMAssay Description:Binding affinity to wild type His-tagged STING (unknown origin) measured after 3 hrs incubation by HTRF assayMore data for this Ligand-Target Pair





3D Structure (crystal)















